SCHEMBL7446091

SCHEMBL7446091

O=CCn1c(-c2ccc(F)cc2)ccc(NC(=O)OCc2ccccc2)c1=O

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ELANE P08246 18/20 0.53
CTRC Q99895 3/20 0.53
MGLL Q99685 1/20 0.49
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7283751 0.93 ELANE (0.57) ELANECTRCMGLLNPC1RAB9A
SCHEMBL8536676 0.88 ELANE (0.59) ELANECTRCMGLL
SCHEMBL7440440 0.83 ELANE (0.55) ELANECTRCMGLL
SCHEMBL7276667 0.83 ELANE (0.62) ELANECTRC
SCHEMBL6558159 0.83 ELANE (0.63) ELANEMGLL
SCHEMBL7445689 0.82 ELANE (0.60) ELANECTRCNPC1RAB9A
SCHEMBL7284545 0.81 HDAC3 (0.52) ELANECTRCNPC1RAB9A
SCHEMBL7274908 0.81 POLB (0.44) ELANECTRCNPC1RAB9A
SCHEMBL7276488 0.79 ELANE (0.64) ELANECTRCNPC1RAB9A
SCHEMBL7300356 0.76 ELANE (0.61) ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636142-B1 LACTAM PEPTIDES HAVING HLE INHIBITING ACTIVITY ZENECA LTD (GB) 1998-06-17 EP disclosed
US-5721222-A Heterocyclic ketones ZENECA LIMITED (GB) 1998-02-24 US disclosed
US-5486529-A Certain pyridyl ketones for treating diseases involving leukocyte elastase ZENECA LIMITED (GB) 1996-01-23 US disclosed
EP-0636142-A1 LACTAM PEPTIDES HAVING HLE INHIBITING ACTIVITY ZENECA LIMITED (GB) 1995-02-01 EP disclosed
WO-1993021209-A1 LACTAM PEPTIDES HAVING HLE INHIBITING ACTIVITY ZENECA LIMITED (GB) 1993-10-28 WO disclosed