SCHEMBL7446291

SCHEMBL7446291

CSc1nc(N)cc(=O)n1Cc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.50
BRAF P15056 1/20 0.49
NPSR1 Q6W5P4 1/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
CYP3A4 P08684 1/20 0.47
DHFR P00374 6/20 0.46
POLB P06746 1/20 0.45
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TLR7 Q9NYK1 1/20 0.43
TSHR P16473 1/20 0.43
HTT P42858 1/20 0.43
TYMS P04818 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26790950 0.74 BRAF (0.61) HPGDBRAFNPSR1MEN1KMT2A
SCHEMBL5025892 0.72 LMNA (0.66) MEN1KMT2ACYP3A4DHFRPOLB
SCHEMBL11841190 0.71 P2RX4 (0.58) HPGDBRAFNPSR1MEN1KMT2A
SCHEMBL10634597 0.71 NPC1 (0.47) BRAFNPSR1MEN1KMT2ADHFR
SCHEMBL11699978 0.71 CYP3A4 (0.55) HPGDCYP3A4POLBALDH1A1TLR7
SCHEMBL13325137 0.70 ALDH1A1 (0.52) HPGDMEN1KMT2AKDM4EALDH1A1
SCHEMBL18931751 0.70 HPGD (0.51) HPGDMEN1KMT2ACYP3A4POLB
SCHEMBL9409123 0.70 SCN5A (0.51) HPGDKMT2APOLBKDM4EALDH1A1
SCHEMBL1227299 0.70 MAP4K1 (0.48) HPGDNPSR1MEN1KMT2ACYP3A4
SCHEMBL19468886 0.69 BACE1 (0.51) HPGDMEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0538332-B1 POLYCYCLIC GUANINE DERIVATIVES SCHERING CORP (US) 1997-07-23 EP disclosed
US-5393755-A Hypotensive agents, enzyme inhibitors SCHERING CORPORATION (US) 1995-02-28 US disclosed
EP-0538332-A1 POLYCYCLIC GUANINE DERIVATIVES. SCHERING CORP (US) 1993-04-28 EP disclosed
WO-1991019717-A1 POLYCYCLIC GUANINE DERIVATIVES SCHERING CORPORATION (US) 1991-12-26 WO disclosed