SCHEMBL7446408

SCHEMBL7446408

CC(=O)Oc1ccc2c(c1OC(C)=O)CC(c1ccccc1)C=C2CNC(=O)OC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.35
KDM4A O75164 1/20 0.34
PTPN1 P18031 2/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
NAMPT P43490 1/20 0.33
HDAC1 Q13547 1/20 0.33
KDM1A O60341 1/20 0.33
MAOB P27338 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4E B2RXH2 3/20 0.33
LMNA P02545 2/20 0.33
HPGD P15428 2/20 0.33
ACACB O00763 2/20 0.33
ACACA Q13085 2/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7447474 0.99 DRD2 (0.35) DRD2KDM4APTPN1ADORA3ADORA2A
SCHEMBL7447921 0.90 KMT2A (0.38) KMT2A
SCHEMBL7447927 0.90 KMT2A (0.38) KMT2A
SCHEMBL7315264 0.90 KDM4A (0.36) DRD2KDM4ANAMPTHDAC1KDM1A
Hydrochloric Acid SCHEMBL7440751 0.89 KMT2A (0.37) KMT2A
SCHEMBL7443351 0.89 ADORA3 (0.36) DRD2PTPN1ADORA3ADORA2AADORA1
SCHEMBL7444847 0.84 CARM1 (0.36) DRD2PTPN1ADORA3ADORA2AADORA1
SCHEMBL7444849 0.84 CARM1 (0.36) DRD2PTPN1ADORA3ADORA2AADORA1
SCHEMBL9038396 0.82 PTPN1 (0.37) DRD2PTPN1ADORA3ADORA2AADORA1
Hydrochloric Acid SCHEMBL8829320 0.82 MASP2 (0.33) HDAC1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5621133-A PREPARING A 1-(3,4-DIALKOXYPHENYL),3-HYDROXYALKANE(C6-C12) BY EPOXIDIZING A HALO DERIVATIVE WITH A BASE FOLLOWED BY DECYCLICIZING WITH AN ORGANOMETALLIC COMPOUND IN A SOLVENT; NAPHTHYLENES, ISOCHROMENES AND ISOTHIOCHROMENES DENINNO MICHAEL P (US) 1997-04-15 US disclosed
US-5591884-A PROTECTED HYDROXYALKYLCATECHOL INTERMEDIATES ABBOTT LABORATORIES (US) 1997-01-07 US disclosed
WO-1996038435-A1 DOPAMINE AGONISTS ABBOTT LABORATORIES (US) 1996-12-05 WO disclosed
EP-0474767-B1 DOPAMINE AGONISTS ABBOTT LAB (US) 1996-02-21 EP disclosed
EP-0474767-A4 DOPAMINE AGONISTS 1992-07-08 EP disclosed
EP-0474767-A1 DOPAMINE AGONISTS. ABBOTT LAB (US) 1992-03-18 EP disclosed
WO-1990015056-A1 DOPAMINE AGONISTS ABBOTT LABORATORIES (US) 1990-12-13 WO disclosed