Benzene

Benzene

SCHEMBL7447284

COC(=O)c1ccc(NC(=O)c2ccccc2C)c(OC)c1.c1ccccc1

nearest known ligand 0.70

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.70
PYGL P06737 4/20 0.61
KMT2A Q03164 5/20 0.54
POLB P06746 2/20 0.54
KCNK3 O14649 1/20 0.54
KCNK9 Q9NPC2 1/20 0.54
MAPT P10636 4/20 0.53
MEN1 O00255 3/20 0.53
RAB9A P51151 3/20 0.53
NPC1 O15118 2/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
CHEK1 O14757 1/20 0.53
PIM1 P11309 1/20 0.53
MAPK8 P45983 1/20 0.53
CLK4 Q9HAZ1 1/20 0.53
GAA P10253 3/20 0.53
TP53 P04637 1/20 0.53
MAPK1 P28482 2/20 0.52
HSD17B10 Q99714 2/20 0.52
TSHR P16473 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20601619 0.91 ALDH1A1 (0.72) ALDH1A1PYGLKMT2APOLBKCNK3
SCHEMBL31586318 0.91 ALDH1A1 (0.72) ALDH1A1PYGLKMT2APOLBKCNK3
SCHEMBL7343390 0.86 KMT2A (0.72) ALDH1A1PYGLKMT2AMAPTMEN1
SCHEMBL5316685 0.85 HTT (0.59) ALDH1A1PYGLKMT2APOLBMAPT
SCHEMBL5233294 0.84 ALDH1A1 (0.56) ALDH1A1PYGLKMT2AMAPTMEN1
SCHEMBL7344448 0.82 PYGL (0.58) ALDH1A1PYGLKMT2AMAPTMEN1
SCHEMBL7339795 0.81 SGMS2 (0.57) ALDH1A1PYGLKMT2AMAPTMEN1
SCHEMBL11784909 0.81 KMT2A (0.72) ALDH1A1KMT2APOLBKCNK3KCNK9
SCHEMBL16147709 0.79 PYGL (0.55) ALDH1A1PYGLKMT2AMAPTMEN1
SCHEMBL4777763 0.79 MAPT (0.51) ALDH1A1PYGLKMT2APOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915876-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS American Cyanamid Company (US) 1999-05-19 EP disclosed
WO-1997049708-A9 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS 1998-05-22 WO disclosed
WO-1997049707-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1997-12-31 WO disclosed
EP-0804438-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS American Cyanamid Company (US) 1997-11-05 EP disclosed
EP-0804440-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS American Cyanamid Company (US) 1997-11-05 EP disclosed
WO-1996022295-A9 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS 1996-11-14 WO disclosed
WO-1996022295-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1996-07-25 WO disclosed