SCHEMBL16147709

SCHEMBL16147709

COC(=O)c1ccc(NC(=O)c2cccc(Cl)c2O)c(OC)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYGL P06737 2/20 0.55
HDAC1 Q13547 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
KMT2A Q03164 4/20 0.52
KDM4E B2RXH2 4/20 0.52
ALDH1A1 P00352 2/20 0.52
TOP1 P11387 1/20 0.52
PDE4D Q08499 1/20 0.51
NPC1 O15118 6/20 0.50
RAB9A P51151 5/20 0.50
SMN1; SMN2 Q16637 5/20 0.50
MEN1 O00255 3/20 0.50
MAPT P10636 3/20 0.50
LMNA P02545 2/20 0.50
GRM4 Q14833 2/20 0.50
NPSR1 Q6W5P4 2/20 0.50
MAPK1 P28482 1/20 0.49
NOD2 Q9HC29 1/20 0.49
WDR5 P61964 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7343390 0.83 KMT2A (0.72) PYGLKMT2AKDM4EALDH1A1NPC1
SCHEMBL16147456 0.80 KCNMA1 (0.67) PYGLHDAC1HDAC8HDAC6KMT2A
SCHEMBL20601819 0.79 WDR5 (0.54) PYGLHDAC1HDAC8HDAC6KMT2A
SCHEMBL20601662 0.79 PYGL (0.82) PYGLHDAC1HDAC8HDAC6KMT2A
Benzene SCHEMBL7447284 0.79 ALDH1A1 (0.70) PYGLKMT2AKDM4EALDH1A1NPC1
SCHEMBL3134272 0.79 ALDH1A1 (0.58) PYGLHDAC8KMT2AKDM4EALDH1A1
SCHEMBL16392552 0.78 PYGL (0.48) PYGLHDAC1KMT2AKDM4EALDH1A1
SCHEMBL5316685 0.77 HTT (0.59) PYGLKMT2AKDM4EALDH1A1NPC1
SCHEMBL7344448 0.77 PYGL (0.58) PYGLKMT2AALDH1A1TOP1NPC1
SCHEMBL5233294 0.77 ALDH1A1 (0.56) PYGLKMT2AKDM4EALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014165816-A1 COMPOUNDS USEFUL FOR THE TREATMENT OF METABOLIC DISORDERS AND SYNTHESIS OF THE SAME NORTH CAROLINA CENTRAL UNIVERSITY (US) 2014-10-09 WO disclosed