SCHEMBL7447552

SCHEMBL7447552

COC(=O)C(CCc1ccccc1)NS(=O)(=O)N1CCN(c2ccc(Cl)cn2)CC1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 8/20 0.43
HDAC2 Q92769 2/20 0.43
HDAC3 O15379 1/20 0.43
CYP2C9 P11712 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
MAPKAPK3 Q16644 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
CHRM4 P08173 2/20 0.40
CHRM2 P08172 3/20 0.39
CHRM1 P11229 3/20 0.39
ALDH1A1 P00352 3/20 0.39
RAB9A P51151 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
NPC1 O15118 2/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 2/20 0.39
HTT P42858 2/20 0.39
TP53 P04637 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4677805 0.87 DRD4 (0.42) ALDH1A1RAB9ASMN1; SMN2NPC1MAPT
SCHEMBL4677803 0.87 DRD4 (0.42) ALDH1A1RAB9ASMN1; SMN2NPC1MAPT
SCHEMBL4673472 0.73 RORC (0.42) ALDH1A1RAB9ASMN1; SMN2NPC1MAPT
SCHEMBL4673464 0.73 RORC (0.42) ALDH1A1RAB9ASMN1; SMN2NPC1MAPT
SCHEMBL4813294 0.67 DRD2 (0.42) ALDH1A1MAPTKDM4EDRD4TSHR
SCHEMBL4673431 0.67 RORC (0.42) HDAC8ALDH1A1RAB9ASMN1; SMN2NPC1
SCHEMBL4673423 0.67 RORC (0.42) HDAC8ALDH1A1RAB9ASMN1; SMN2NPC1
SCHEMBL4671050 0.66 MMP1 (0.52) CHRM1RAB9ADRD4DRD2
SCHEMBL4671045 0.66 MMP1 (0.52) CHRM1RAB9ADRD4DRD2
SCHEMBL16938448 0.65 CA2 (0.48) CYP2C9ALDH1A1RAB9ASMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0958287-A1 SULFAMIDE-METALLOPROTEASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 1999-11-24 EP disclosed
WO-1998032748-A1 SULFAMIDE-METALLOPROTEASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 1998-07-30 WO disclosed