SCHEMBL7447623

SCHEMBL7447623

COC(=O)CC(CC(=O)O)c1cccc(F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
KDM4E B2RXH2 1/20 0.46
F2 P00734 4/20 0.44
F10 P00742 4/20 0.44
MAPT P10636 2/20 0.44
FNTA P49354 1/20 0.44
FNTB P49356 1/20 0.44
POLB P06746 1/20 0.44
MAPK1 P28482 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
CNR2 P34972 1/20 0.44
PRSS1 P07477 3/20 0.44
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
ALOX15 P16050 1/20 0.43
CYP2C19 P33261 1/20 0.43
CYP26A1 O43174 1/20 0.43
FFAR1 O14842 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5857867 0.88 GABBR2 (0.50) MAPTFNTAFNTBHDAC4HDAC7
SCHEMBL12268202 0.83 ALDH1A1 (0.61) ALDH1A1KDM4EMAPTFNTAFNTB
SCHEMBL1811811 0.83 ALDH1A1 (0.61) ALDH1A1KDM4EMAPTFNTAFNTB
SCHEMBL14691022 0.83 FNTA (0.51) ALDH1A1F2F10MAPTFNTA
SCHEMBL27788467 0.82 FFAR1 (0.46) HDAC4HDAC7HDAC5CNR2CYP26A1
SCHEMBL6581023 0.82 ALDH1A1 (0.55) ALDH1A1MAPTFNTAFNTBCYP2D6
SCHEMBL6581020 0.82 ALDH1A1 (0.55) ALDH1A1MAPTFNTAFNTBCYP2D6
SCHEMBL6581305 0.82 ALDH1A1 (0.55) ALDH1A1MAPTFNTAFNTBCYP2D6
SCHEMBL7682611 0.81 F2 (0.41) ALDH1A1KDM4EF2F10MAPT
SCHEMBL8770903 0.81 L3MBTL1 (0.49) ALDH1A1KDM4EMAPTPOLBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1105389-A4 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2001-10-17 EP disclosed
EP-1105389-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2001-06-13 EP disclosed
US-6090944-A Alkanoic acid derivatives as αv integrin receptor antagonists MERCK & CO., INC. (US) 2000-07-18 US disclosed
WO-2000009503-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2000-02-24 WO disclosed