SCHEMBL7447640

SCHEMBL7447640

CCCC(=O)c1ccc(Cl)cc1N

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.56
TSHR P16473 3/20 0.51
NOS2 P35228 2/20 0.50
ALDH1A1 P00352 7/20 0.44
ALOX15 P16050 4/20 0.44
TDP1 Q9NUW8 3/20 0.44
RECQL P46063 2/20 0.44
HPGD P15428 2/20 0.44
HSD17B10 Q99714 2/20 0.44
FLT1 P17948 1/20 0.44
FLT4 P35916 1/20 0.44
KDR P35968 1/20 0.44
POLB P06746 2/20 0.44
THRB P10828 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
MAPK1 P28482 2/20 0.43
HIF1A Q16665 1/20 0.43
GAA P10253 1/20 0.43
PKM P14618 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2081805 0.86 NOS2 (0.65) ABL1TSHRNOS2ALDH1A1ALOX15
SCHEMBL9041985 0.86 ABL1 (0.59) ABL1TSHRNOS2ALDH1A1ALOX15
SCHEMBL30249612 0.86 ABL1 (0.59) ABL1TSHRNOS2ALDH1A1ALOX15
SCHEMBL18637905 0.83 ABL1 (0.51) ABL1TSHRNOS2ALDH1A1HPGD
SCHEMBL27439105 0.83 ABL1 (0.51) ABL1TSHRNOS2ALDH1A1ALOX15
SCHEMBL2125979 0.82 ALDH1A1 (0.65) TSHRALDH1A1ALOX15TDP1RECQL
SCHEMBL5636998 0.81 ABL1 (0.50) ABL1TSHRNOS2ALDH1A1ALOX15
SCHEMBL18758662 0.81 ABL1 (0.62) ABL1NOS2ALDH1A1HSD17B10FLT1
SCHEMBL11230620 0.81 TSHR (0.52) TSHRNOS2ALDH1A1ALOX15TDP1
SCHEMBL7965902 0.81 ALDH1A1 (0.59) TSHRNOS2ALDH1A1ALOX15TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189905-A1 SUBSTITUTED HETEROCYCLE FUSED GAMMA-CARBOLINES Bristol-Myers Squibb Pharma Company (US) 2002-03-27 EP disclosed
WO-2000077001-A1 SUBSTITUTED HETEROCYCLE FUSED GAMMA-CARBOLINES DU PONT PHARMACEUTICALS COMPANY (US) 2000-12-21 WO disclosed
EP-0325247-B1 CAMPTOTHECIN DERIVATIVES AND PROCESS FOR PREPARING SAME KABUSHIKI KAISHA YAKULT HONSHA (JP) 1993-05-19 EP disclosed
US-5061800-A ANTITUMOR AGENTS KABUSHIKI KAISHA YAKULT HONSHA (JP) 1991-10-29 US disclosed
EP-0325247-A1 Camptothecin derivatives and process for preparing same KABUSHIKI KAISHA YAKULT HONSHA (JP) 1989-07-26 EP disclosed