SCHEMBL7447670

SCHEMBL7447670

Cc1ccc(S(=O)(=O)N(C(=O)[C@H]2NC(C)(C)CS2)[C@@H](Cc2ccc(OCCN(C)C)cc2)C(=O)O)cc1.Cc1ccc(S(=O)(=O)N2CCC[C@H]2C(=O)N[C@@H](Cc2ccc(OCCN(C)C)cc2)C(=O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 4/20 0.46
ITGB1 P05556 8/20 0.43
ITGA5 P08648 3/20 0.43
ITGB7 P26010 1/20 0.41
ITGAV P06756 3/20 0.39
ALDH1A1 P00352 1/20 0.39
ITGA2 P17301 1/20 0.38
KCNQ1 P51787 3/20 0.37
KMT2A Q03164 1/20 0.36
FKBP1A P62942 1/20 0.36
MMP1 P03956 1/20 0.36
ADAM17 P78536 1/20 0.36
TSHR P16473 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7319946 0.86 KMT2A (0.35) ALDH1A1KMT2AADAM17
SCHEMBL7446810 0.85 ITGB1 (0.51) ITGA4ITGB1ITGA5ITGAVALDH1A1
SCHEMBL7325150 0.85 ITGA4 (0.60) ITGA4ITGB1ITGA5ITGB7ITGAV
SCHEMBL7449470 0.85 ITGB1 (0.48) ITGA4ITGB1ITGA5ITGAVALDH1A1
SCHEMBL7314611 0.83 ITGB3 (0.35) ALDH1A1KMT2A
SCHEMBL7315770 0.81 ITGA4 (0.59) ITGA4ITGB1ITGA5ITGB7ITGAV
SCHEMBL7319858 0.79 ITGA4 (0.59) ITGA4ITGB1ITGA5ITGB7ITGAV
SCHEMBL7322201 0.78 ITGA4 (0.60) ITGA4ITGB1ITGA5ITGB7ITGAV
SCHEMBL5609014 0.77 ITGB1 (0.39) ITGA4ITGB1ITGA5ITGB7ITGAV
SCHEMBL7318412 0.76 ALDH1A1 (0.37) ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001972-A1 SUBSTITUTED PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-05-24 EP claimed
WO-1999006431-A1 SUBSTITUTED PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO claimed