SCHEMBL7448164

SCHEMBL7448164

CCN(Cc1cc(O)c(C(c2cccc(NS(=O)(=O)c3cc(Cl)ccc3Cl)c2)C2CC2)c(=O)o1)S(=O)(=O)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
LMNA P02545 3/20 0.40
MAPT P10636 3/20 0.38
HTT P42858 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HSP90AA1 P07900 5/20 0.37
HSP90AB1 P08238 5/20 0.37
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HSD11B1 P28845 1/20 0.34
TP53 P04637 1/20 0.34
ITGA1 P56199 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
KDM4E B2RXH2 1/20 0.33
AR P10275 1/20 0.33
RAB9A P51151 1/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7441056 0.90 ALDH1A1 (0.40) ALDH1A1LMNAMAPTHTTL3MBTL1
Ethane SCHEMBL7485196 0.87 HSP90AA1 (0.39) ALDH1A1LMNAMAPTHTTTDP1
SCHEMBL7450446 0.86 ALDH1A1 (0.42) ALDH1A1LMNAMAPTHTTHSP90AA1
SCHEMBL7432830 0.85 PTGER2 (0.37) ALDH1A1LMNAMAPTHTTMEN1
SCHEMBL7437314 0.85 ALDH1A1 (0.38) ALDH1A1LMNAMAPTHTTL3MBTL1
SCHEMBL7444165 0.85 PDE4B (0.40) ALDH1A1LMNAMAPTHTTTDP1
SCHEMBL7437641 0.84 LMNA (0.38) ALDH1A1LMNAMAPTHTTMEN1
SCHEMBL7445404 0.83 PARP1 (0.37) ALDH1A1LMNAMAPTHTTL3MBTL1
SCHEMBL7445970 0.83 ALDH1A1 (0.37) ALDH1A1LMNAMAPTHTTTDP1
SCHEMBL7448174 0.82 HSP90AA1 (0.38) ALDH1A1LMNAMAPTHTTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
EP-1203770-A1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases PHARMACIA & UPJOHN COMPANY (US) 2002-05-08 EP disclosed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed