SCHEMBL7448201

SCHEMBL7448201

Cc1c(CNC(=O)N2CCCC2)ccc2[nH]c(CNc3ccc(C#N)cc3)nc12

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.39
MLLT1 Q03111 1/20 0.39
TGFBR1 P36897 4/20 0.37
DGAT2 Q96PD7 3/20 0.37
IDH1 O75874 2/20 0.36
OPRM1 P35372 1/20 0.35
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPK1 P28482 1/20 0.34
RAB9A P51151 1/20 0.34
KIT P10721 1/20 0.34
MAPK14 Q16539 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
CSNK1E P49674 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PANK3 Q9H999 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7449699 0.81 MLLT1 (0.38) MLLT1TGFBR1DGAT2IDH1OPRM1
SCHEMBL7442673 0.76 MLLT1 (0.34) MLLT1TGFBR1DGAT2IDH1OPRM1
SCHEMBL7446445 0.75 NPC1 (0.38) MLLT1TGFBR1DGAT2IDH1LMNA
SCHEMBL7454489 0.75 NPC1 (0.38) MLLT1TGFBR1DGAT2IDH1LMNA
SCHEMBL7447505 0.75 NPC1 (0.36) MLLT1TGFBR1DGAT2IDH1LMNA
SCHEMBL7447136 0.74 ALDH1A1 (0.37) MLLT1TGFBR1DGAT2IDH1LMNA
SCHEMBL6455288 0.74 MLLT1 (0.33) MLLT1TGFBR1DGAT2
SCHEMBL7421109 0.74 NPC1 (0.37) MLLT1TGFBR1DGAT2IDH1LMNA
SCHEMBL7445643 0.72 NPC1 (0.35) MLLT1TGFBR1DGAT2LMNAMAPT
Hydrochloric Acid SCHEMBL7446984 0.71 KLK1 (0.40) LMNAMAPTNPC1ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095025-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM KG (DE) 2001-05-02 EP disclosed
WO-2000001704-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-01-13 WO disclosed