SCHEMBL7448284

SCHEMBL7448284

O=C(O)C[C@H](NS(=O)(=O)c1cc(Cl)cc(Cl)c1)C(=O)N[C@@H](Cc1ccc(F)cc1)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.49
ITGA4 P13612 1/20 0.49
CA2 P00918 2/20 0.47
MMP2 P08253 5/20 0.46
ADAMTS5 Q9UNA0 1/20 0.46
ACE P12821 1/20 0.46
EEF2K O00418 1/20 0.43
ALDH1A1 P00352 1/20 0.42
MMP9 P14780 3/20 0.42
ADAMTS4 O75173 1/20 0.42
L3MBTL1 Q9Y468 3/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
TDP1 Q9NUW8 1/20 0.41
POLB P06746 1/20 0.41
MME P08473 1/20 0.41
CTSB P07858 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7442952 0.94 ITGB1 (0.53) ITGB1ITGA4CA2MMP2ADAMTS5
SCHEMBL7448892 0.92 MMP2 (0.53) ITGB1ITGA4CA2MMP2ADAMTS5
SCHEMBL7444227 0.91 ITGB1 (0.55) ITGB1ITGA4CA2MMP2ADAMTS5
SCHEMBL7453817 0.90 ITGB1 (0.49) ITGB1ITGA4CA2MMP2ADAMTS5
SCHEMBL7453591 0.90 MEN1 (0.52) ITGB1ITGA4CA2MMP2ADAMTS5
SCHEMBL7447697 0.86 ITGB1 (0.46) ITGB1ITGA4CA2MMP2ADAMTS5
SCHEMBL7450515 0.85 CA2 (0.50) ITGB1ITGA4CA2MMP2ADAMTS5
SCHEMBL7446008 0.84 GPR132 (0.50) ITGB1ITGA4CA2MMP2ADAMTS5
SCHEMBL7450626 0.83 ITGB1 (0.48) ITGB1ITGA4CA2MMP2ADAMTS5
SCHEMBL7447633 0.77 CTSL (0.50) MMP2ALDH1A1MMP9MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6221888-B1 ANTIHISTAMINE, ANTIINFLAMMATORY AGENT, AUTOIMMUNE DISEASE, RHEUMATIC DISORDERS MERCK & CO., INC. 2001-04-24 US claimed
EP-0998282-A4 SULFONAMIDES AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2000-08-30 EP claimed
EP-0998282-A1 SULFONAMIDES AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-10 EP claimed
WO-1998053818-A1 SULFONAMIDES AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed