SCHEMBL7448296

SCHEMBL7448296

Cc1ccc(S(=O)(=O)N2CCC[C@H]2C(=O)N[C@@H](CCC(=O)NCCc2[nH]ccc2C)C(=O)O)cc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.50
TP53 P04637 1/20 0.50
CASP1 P29466 1/20 0.50
CASP7 P55210 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
HSD17B10 Q99714 1/20 0.50
FKBP1A P62942 2/20 0.49
ITGA4 P13612 2/20 0.47
ITGB1 P05556 4/20 0.46
ITGA2 P17301 1/20 0.46
ITGA5 P08648 3/20 0.45
GAA P10253 1/20 0.44
HPGD P15428 1/20 0.44
L3MBTL1 Q9Y468 3/20 0.44
RAB9A P51151 1/20 0.42
MAPK1 P28482 1/20 0.42
ITGAV P06756 1/20 0.42
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5492997 0.84 FKBP1A (0.57) LMNATP53CASP1CASP7SMN1; SMN2
SCHEMBL5497978 0.83 FKBP1A (0.52) LMNATP53CASP1CASP7SMN1; SMN2
SCHEMBL5499031 0.83 LMNA (0.57) LMNATP53CASP1CASP7SMN1; SMN2
SCHEMBL6709564 0.81 ITGA4 (0.57) FKBP1AITGA4ITGB1ITGA2ITGA5
SCHEMBL6710636 0.81 ITGA4 (0.57) FKBP1AITGA4ITGB1ITGA2ITGA5
SCHEMBL5496192 0.80 ITGA4 (0.56) FKBP1AITGA4ITGB1ITGA2ITGA5
SCHEMBL6151165 0.78 ITGA4 (0.58) FKBP1AITGA4ITGB1ITGA2ITGA5
SCHEMBL6151162 0.78 ITGA4 (0.58) FKBP1AITGA4ITGB1ITGA2ITGA5
SCHEMBL5494189 0.78 FKBP1A (0.67) LMNATP53CASP1CASP7SMN1; SMN2
SCHEMBL6710949 0.77 GAA (0.60) FKBP1AITGA4ITGB1ITGA2ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001971-A1 DIPEPTIDE AND RELATED COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-05-24 EP claimed
WO-1999006432-A1 DIPEPTIDE AND RELATED COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO claimed
EP-1001971-A1 DIPEPTIDE AND RELATED COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-05-24 EP disclosed
WO-1999006432-A1 DIPEPTIDE AND RELATED COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO disclosed