SCHEMBL7448750

SCHEMBL7448750

CCOC(=O)CCN(C(=O)Oc1ccc2[nH]c(CNc3ccc(C#N)cc3)nc2c1C)C1CCCC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 2/20 0.36
PDE3B Q13370 2/20 0.36
PDE3A Q14432 2/20 0.36
P2RY12 Q9H244 2/20 0.36
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 1/20 0.35
PYGL P06737 1/20 0.34
PIP4K2A P48426 1/20 0.32
KDM4E B2RXH2 3/20 0.32
TGFBR1 P36897 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7453833 0.89 PDE3B (0.36) PDE2APDE3BPDE3AP2RY12ALDH1A1
Hydrochloric Acid SCHEMBL7448617 0.88 KLK1 (0.41) PDE2APDE3BPDE3AP2RY12ALDH1A1
SCHEMBL7453272 0.80 KLK1 (0.43) ALDH1A1MAPTNPC1LMNAMAPK1
SCHEMBL7449392 0.80 NPC1 (0.34) ALDH1A1MAPTNPC1LMNAMAPK1
SCHEMBL7444335 0.79 MAPT (0.41) ALDH1A1MAPTNPC1LMNAMAPK1
Hydrochloric Acid SCHEMBL7449551 0.77 PDE3B (0.36) PDE2APDE3BPDE3AP2RY12MAPT
SCHEMBL7445637 0.77 ALDH1A1 (0.39) ALDH1A1MAPTNPC1LMNAMAPK1
SCHEMBL7451792 0.74 IDH1 (0.39) ALDH1A1MAPTNPC1LMNAMAPK1
Hydrochloric Acid SCHEMBL7445965 0.73 KLK1 (0.41) ALDH1A1MAPTNPC1LMNAMAPK1
SCHEMBL9901721 0.73 NQO2 (0.46) ALDH1A1MAPTNPC1LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966454-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS Boehringer Ingelheim Pharma KG (DE) 1999-12-29 EP disclosed
WO-1998037075-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1998-08-27 WO disclosed