SCHEMBL7450449

SCHEMBL7450449

CCC(NS(=O)(=O)c1ccccc1)c1cc(O)c(C(c2cccc(NS(=O)(=O)c3ccc(F)cc3)c2)C2CC2)c(=O)o1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
KCNA5 P22460 1/20 0.36
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
HSD17B3 P37058 1/20 0.36
HSD17B2 P37059 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4D Q08499 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ATM Q13315 1/20 0.35
ALOX12 P18054 1/20 0.35
KCNK3 O14649 2/20 0.34
LIMK2 P53671 1/20 0.34
RORC P51449 1/20 0.34
MMP12 P39900 1/20 0.34
MMP13 P45452 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7441063 0.95 KCNK3 (0.36) KCNA5PDE4BALOX12KCNK3MMP12
SCHEMBL7437319 0.91 ALDH1A1 (0.36) ALOX12KCNK3LIMK2MMP12MMP13
SCHEMBL7437644 0.90 EEF2K (0.41) HSD17B2
SCHEMBL7442097 0.89 ATM (0.37) MEN1KMT2AHSP90AA1HSP90AB1HSD17B3
SCHEMBL7447436 0.87 LIMK2 (0.37) MEN1KMT2AKCNA5HSP90AA1HSP90AB1
SCHEMBL7445975 0.87 POLB (0.38) KMT2AKCNA5L3MBTL1ATM
SCHEMBL7448174 0.86 HSP90AA1 (0.38) MEN1KMT2AHSP90AA1HSP90AB1PDE4B
Ethane SCHEMBL7484090 0.84 ALOX12 (0.38) MEN1KMT2AHSP90AA1HSP90AB1HSD17B3
SCHEMBL7443310 0.84 POLB (0.36) ALOX12
SCHEMBL7405143 0.83 HSD17B2 (0.39) MEN1KMT2AHSP90AA1HSP90AB1HSD17B3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO claimed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed