SCHEMBL7451127

SCHEMBL7451127

O=C(Nc1ccnc(Cl)c1)c1nc(C2CC2)n2c1CSc1ccccc1-2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.45
SMARCA2 P51531 7/20 0.37
SMARCA4 P51532 6/20 0.37
JAK2 O60674 3/20 0.34
TYK2 P29597 3/20 0.34
JAK1 P23458 2/20 0.34
PRKCI P41743 1/20 0.34
CDK9 P50750 1/20 0.34
JAK3 P52333 1/20 0.34
HDAC4 P56524 1/20 0.33
PIK3CA P42336 1/20 0.33
MTOR P42345 1/20 0.33
PIK3CG P48736 1/20 0.33
NPC1 O15118 1/20 0.33
USP2 O75604 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7451341 0.86 GRM5 (0.53) GRM5SMARCA2SMARCA4NPC1USP2
SCHEMBL7453227 0.84 GRM5 (0.47) GRM5SMARCA2SMARCA4HDAC4MAPT
SCHEMBL7454592 0.78 GRM5 (0.68) GRM5SMARCA2SMARCA4NPC1USP2
SCHEMBL7454850 0.78 GRM5 (0.52) GRM5SMARCA2SMARCA4NPC1USP2
SCHEMBL7449902 0.77 GRM5 (0.46) GRM5SMARCA2SMARCA4NPC1USP2
SCHEMBL7446764 0.76 GRM5 (0.52) GRM5SMARCA2SMARCA4NPC1MAPT
SCHEMBL7451159 0.74 GRM5 (0.60) GRM5SMARCA2SMARCA4
SCHEMBL7451577 0.74 GRM5 (0.55) GRM5SMARCA2SMARCA4HDAC4NPC1
SCHEMBL12067831 0.72 L3MBTL1 (0.45) NPC1LMNATP53MAPTHTT
SCHEMBL7447799 0.71 GRM5 (0.44) GRM5SMARCA2SMARCA4NPC1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011151361-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2011-12-08 WO claimed
WO-2011151361-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2011-12-08 WO disclosed
WO-2011151361-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2011-12-08 WO disclosed