SCHEMBL7452192

SCHEMBL7452192

Cc1c(OC(=O)N(CCCC(=O)OC(C)(C)C)c2ccccc2)ccc2[nH]c(CNc3ccc(C#N)cc3)nc12

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34
RAB9A P51151 1/20 0.34
CYP1A2 P05177 1/20 0.32
TSHR P16473 1/20 0.32
CHRM2 P08172 2/20 0.32
CHRM1 P11229 2/20 0.32
CHRM3 P20309 2/20 0.32
TGFBR1 P36897 2/20 0.31
TNKS O95271 1/20 0.31
PARP1 P09874 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
F2 P00734 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7444335 0.85 MAPT (0.41) NPC1ALDH1A1LMNAMAPTMAPK1
Hydrochloric Acid SCHEMBL7441375 0.79 F2 (0.43) NPC1ALDH1A1LMNAMAPTMAPK1
SCHEMBL7445168 0.79 F2 (0.51) NPC1ALDH1A1LMNAMAPTMAPK1
Hydrochloric Acid SCHEMBL7449253 0.78 F2 (0.50) NPC1ALDH1A1LMNAMAPTMAPK1
SCHEMBL7451792 0.77 IDH1 (0.39) NPC1ALDH1A1LMNAMAPTMAPK1
SCHEMBL7441087 0.77 SMN1; SMN2 (0.35) NPC1ALDH1A1LMNAMAPTMAPK1
SCHEMBL7453241 0.77 F2 (0.48) NPC1ALDH1A1LMNAMAPTMAPK1
Hydrochloric Acid SCHEMBL7452868 0.77 KLK1 (0.45) NPC1ALDH1A1LMNAMAPTMAPK1
Hydrochloric Acid SCHEMBL7449067 0.77 KLK1 (0.45) NPC1ALDH1A1LMNAMAPTMAPK1
SCHEMBL7445637 0.77 ALDH1A1 (0.39) NPC1ALDH1A1LMNAMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966454-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS Boehringer Ingelheim Pharma KG (DE) 1999-12-29 EP disclosed
WO-1998037075-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1998-08-27 WO disclosed