SCHEMBL7452986

SCHEMBL7452986

[CH2]C(Cc1cccnc1)c1ccccn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.49
CYP1A2 P05177 4/20 0.49
FDPS P14324 1/20 0.44
HTT P42858 2/20 0.41
CHRNA7 P36544 1/20 0.40
LTA4H P09960 1/20 0.39
FNTA P49354 1/20 0.39
FNTB P49356 1/20 0.39
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
CHRNB2 P17787 2/20 0.39
CHRNA4 P43681 2/20 0.39
CYP2A6 P11509 2/20 0.39
CYP3A4 P08684 3/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10871037 0.84 CYP1A2 (0.54) CYP2D6CYP1A2HTTCHRNA7CYP2A6
SCHEMBL5263511 0.81 SLC6A4 (0.42) CYP2D6CYP1A2HTTKDM4ECYP3A4
SCHEMBL7073814 0.81 CYP1A2 (0.49) CYP2D6CYP1A2FDPSHTTCHRNA7
SCHEMBL5191218 0.74 GRIN2D (0.49) FDPSSMN1; SMN2SLC6A2SLC6A4SLC6A3
SCHEMBL4726907 0.72 FDPS (0.56) CYP2D6CYP1A2FDPSCHRNA7KDM4E
SCHEMBL2096123 0.72 FDPS (0.51) CYP2D6CYP1A2FDPSCHRNA7CHRNB2
SCHEMBL9547411 0.71 FDPS (0.59) CYP2D6CYP1A2FDPSCHRNA7KDM4E
SCHEMBL7740273 0.71 CYP2D6 (0.40) CYP2D6CYP1A2FDPSHTTLTA4H
SCHEMBL5454064 0.71 SIGMAR1 (0.44) CYP2D6CYP1A2FDPSRAB9ACYP3A4
SCHEMBL5460636 0.71 CYP19A1 (0.51) CYP2D6CYP1A2FDPSCHRNA7FNTA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1210598-A4 4-UNSUBSTITUTED DIHYDROISOQUINOLINONE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2002-10-30 EP claimed
EP-1210598-A1 4-UNSUBSTITUTED DIHYDROISOQUINOLINONE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION bioscience AG (DE) 2002-06-05 EP claimed
WO-2001014879-A1 4-UNSUBSTITUTED DIHYDROISOQUINOLINONE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-03-01 WO claimed