SCHEMBL748611

SCHEMBL748611

Cc1ccc(CN(CCc2ccc(Cl)c(Cl)c2)C(=O)c2cccc3c2NCCC3)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.38
MAPT P10636 2/20 0.38
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
TMEM97 Q5BJF2 1/20 0.37
KMT2A Q03164 3/20 0.37
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
ALDH1A1 P00352 2/20 0.36
SIGMAR1 Q99720 7/20 0.34
CYP1A2 P05177 3/20 0.34
CYP2D6 P10635 2/20 0.34
TSHR P16473 2/20 0.34
MEN1 O00255 2/20 0.34
CYP2C19 P33261 1/20 0.34
GRIN2D O15399 1/20 0.34
GRIN3B O60391 1/20 0.34
CYP3A4 P08684 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2A Q12879 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL745501 0.90 TMEM97 (0.39) TP53OPRM1OPRD1TMEM97KMT2A
Hydrochloric Acid SCHEMBL752637 0.90 TMEM97 (0.38) TP53OPRM1OPRD1TMEM97KMT2A
SCHEMBL749603 0.89 TMEM97 (0.39) TP53OPRM1OPRD1TMEM97KMT2A
SCHEMBL749103 0.85 SRC (0.38) TP53MAPTKMT2AALDH1A1SIGMAR1
SCHEMBL746654 0.82 OPRM1 (0.34) TP53MAPTOPRM1OPRD1TMEM97
Hydrochloric Acid SCHEMBL751441 0.82 OPRM1 (0.33) TP53MAPTOPRM1OPRD1TMEM97
SCHEMBL748523 0.81 LPAR1 (0.38) OPRM1OPRD1KMT2ACRHBPCRHR2
SCHEMBL747114 0.80 C5AR1 (0.41) OPRM1OPRD1TMEM97KMT2ACRHBP
SCHEMBL745512 0.80 OPRM1 (0.34) TP53MAPTOPRM1OPRD1TMEM97
SCHEMBL748563 0.79 MBTPS1 (0.39) TP53MAPTOPRM1OPRD1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8022217-B2 Compounds suitable as modulators of HDL CADILA HEALTHCARE LIMITED (IN) 2011-09-20 US claimed
EP-2049493-B1 COMPOUNDS SUITABLE AS MODULATORS OF HDL CADILA HEALTHCARE LTD (IN) 2012-03-21 EP disclosed
US-8022217-B2 Compounds suitable as modulators of HDL CADILA HEALTHCARE LIMITED (IN) 2011-09-20 US disclosed