SCHEMBL7455672

SCHEMBL7455672

O=C(CSCCCc1ccccc1)CSCCCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.54
CA2 P00918 1/20 0.54
MMP12 P39900 1/20 0.54
MMP13 P45452 1/20 0.54
HDAC3 O15379 3/20 0.52
HDAC1 Q13547 3/20 0.52
HDAC2 Q92769 3/20 0.52
HDAC8 Q9BY41 3/20 0.52
HDAC6 Q9UBN7 3/20 0.52
HDAC5 Q9UQL6 3/20 0.52
HDAC4 P56524 2/20 0.52
HDAC7 Q8WUI4 2/20 0.52
HDAC10 Q969S8 2/20 0.52
HDAC11 Q96DB2 2/20 0.52
HDAC9 Q9UKV0 2/20 0.52
MAPK1 P28482 1/20 0.52
ADRA1A P35348 1/20 0.52
SLC6A3 Q01959 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
NOS1 P29475 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5025501 0.89 MMP12 (0.69) CES1CA2MMP12MMP13HDAC3
SCHEMBL709703 0.83 MMP12 (0.67) CES1CA2MMP12MMP13HDAC3
SCHEMBL29308029 0.81 MMP12 (0.65) CES1CA2MMP12MMP13HDAC3
SCHEMBL577035 0.81 CA2 (0.62) CA2HDAC3HDAC1HDAC2HDAC8
SCHEMBL11449287 0.79 ALOX5 (0.52) CES1CA2MMP12MMP13SMN1; SMN2
SCHEMBL4574068 0.78 MMP12 (0.82) CES1CA2MMP12MMP13HDAC3
SCHEMBL708693 0.76 KDM1A (0.51) CES1MMP12MMP13MAPK1SMN1; SMN2
SCHEMBL8990052 0.76 CES1 (0.62) CES1CA2MMP12MMP13HDAC3
SCHEMBL20395222 0.75 CYP2C19 (0.59) SMN1; SMN2MAPTNPC1RAB9ACASP3
SCHEMBL775567 0.74 CYP1A2 (0.58) CA2NOS1MAPTRXFP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1129108-A4 CASPASES AND APOPTOSIS SMITHKLINE BEECHAM CORP (US) 2002-01-09 EP disclosed
EP-1129108-A1 CASPASES AND APOPTOSIS SmithKline Beecham Corporation (US) 2001-09-05 EP disclosed
WO-2000020440-A1 CASPASES AND APOPTOSIS SMITHKLINE BEECHAM CORPORATION (US) 2000-04-13 WO disclosed