SCHEMBL7457264

SCHEMBL7457264

FC(F)(F)c1ccccc1COc1[c]ccc(-c2ccccc2)c1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.45
MAOB P27338 4/20 0.43
MAOA P21397 1/20 0.41
FFAR1 O14842 1/20 0.40
FFAR4 Q5NUL3 1/20 0.40
EPHX2 P34913 2/20 0.38
ADAMTS4 O75173 1/20 0.38
MMP13 P45452 1/20 0.38
SLC6A4 P31645 1/20 0.37
TACR1 P25103 1/20 0.36
AR P10275 1/20 0.35
PTGER4 P35408 1/20 0.35
ALOX5 P09917 1/20 0.35
ALOX5AP P20292 1/20 0.35
MAP4K3 Q8IVH8 1/20 0.35
CHEK1 O14757 1/20 0.35
F2 P00734 1/20 0.34
HCAR2 Q8TDS4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7024874 0.80 IDO1 (0.53) IDO1MAOBMAOAFFAR1FFAR4
SCHEMBL7460676 0.77 KDM4E (0.49) IDO1
SCHEMBL7468357 0.76 AGXT (0.43) IDO1MAOBFFAR1FFAR4ALOX5
SCHEMBL7465277 0.73 AGXT (0.41) IDO1MAOBMAOA
SCHEMBL7470952 0.73 IDO1 (0.45) IDO1MAOBMAOAFFAR1FFAR4
SCHEMBL534316 0.71 PTPN1 (0.37)
SCHEMBL5621755 0.71 RXRA (0.40)
SCHEMBL7464303 0.71 MAOB (0.44) IDO1MAOBMAOAFFAR1
SCHEMBL7464222 0.70 FFAR1 (0.41) IDO1MAOBMAOAFFAR1
SCHEMBL7458294 0.69 AKR1C3 (0.40) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244617-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE Ortho-McNeil Pharmaceutical, Inc. (US) 2002-10-02 EP disclosed
WO-2001047875-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-07-05 WO disclosed