SCHEMBL7459186

SCHEMBL7459186

NCc1ccccc1C(N)=NO

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 6/20 0.47
LMNA P02545 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
GFER P55789 2/20 0.41
PNMT P11086 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.38
MAPT P10636 2/20 0.38
HTT P42858 1/20 0.38
DPP4 P27487 2/20 0.38
ALDH1A1 P00352 2/20 0.34
TAAR1 Q96RJ0 1/20 0.33
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
HTR3A P46098 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32
KDM1A O60341 1/20 0.32
CYP2C19 P33261 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL103625 0.82 GAA (0.46) GAALMNAL3MBTL1GFERSMN1; SMN2
SCHEMBL103624 0.82 GAA (0.46) GAALMNAL3MBTL1GFERSMN1; SMN2
SCHEMBL13770580 0.79 GAA (0.43) GAALMNAL3MBTL1GFERSMN1; SMN2
SCHEMBL21163691 0.77 LMNA (0.44) GAALMNAL3MBTL1GFERSMN1; SMN2
SCHEMBL871585 0.77 BCAT2 (0.51) GAALMNAL3MBTL1MAPTKDM1A
SCHEMBL19153981 0.77 BCAT2 (0.51) GAALMNAL3MBTL1MAPTKDM1A
Water SCHEMBL871348 0.76 BCAT2 (0.50) GAALMNAL3MBTL1MAPTKDM1A
SCHEMBL3188911 0.74 PNMT (0.43) LMNAPNMTSMN1; SMN2HTTDPP4
SCHEMBL405123 0.74 KDM4E (0.52) GAAL3MBTL1PNMTMAPTHTT
SCHEMBL29674786 0.74 PNMT (0.43) LMNAPNMTSMN1; SMN2HTTDPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016201052-A1 BRIDGED BICYCLIC KALLIKREIN INHIBITORS GLOBAL BLOOD THERAPEUTICS, INC. (US) 2016-12-15 WO disclosed
EP-0669317-B1 Prolineamide derivatives MITSUBISHI CHEM CORP (JP) 2002-09-04 EP disclosed
US-5744487-A PROTEASE INHIBITORS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-04-28 US disclosed
EP-0669317-A1 Prolineamide derivatives Mitsubishi Chemical Corporation (JP) 1995-08-30 EP disclosed