SCHEMBL7459503

SCHEMBL7459503

NC(=O)c1nc(-c2ccc(F)cc2)c(CCCl)s1

nearest known ligand 0.43

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 18/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3178699 0.86 GAA (0.48) PTGDR2
SCHEMBL6895646 0.81 PTGS2 (0.58) PTGDR2
SCHEMBL6598899 0.80 PTGDR2 (0.43) PTGDR2
Bromide SCHEMBL6897206 0.77 HTT (0.55) PTGDR2
SCHEMBL3308684 0.76 ALDH1A1 (0.55)
SCHEMBL3185077 0.71 PTGDR2 (0.43) PTGDR2
SCHEMBL8922687 0.71 PTGDR2 (0.46) PTGDR2
SCHEMBL7462975 0.70 TRPM8 (0.47)
SCHEMBL7467556 0.70 HTR2A (0.36) PTGDR2
SCHEMBL27428321 0.69 PTGS2 (0.43) PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0940401-B1 2-CARBONYLTHIAZOLE DERIVATIVES AND USE OF THE SAME TAISHO PHARMACEUTICAL CO LTD (JP) 2002-11-06 EP disclosed
US-6166033-A 2-carbonylthiazole derivatives and use of the same TAISHO PHARMACEUTICAL CO., LTD. (JP) 2000-12-26 US disclosed
EP-0940401-A1 2-CARBONYLTHIAZOLE DERIVATIVES AND USE OF THE SAME TAISHO PHARMACEUTICAL CO. LTD (JP) 1999-09-08 EP disclosed