SCHEMBL7460419

SCHEMBL7460419

O=C(O)C(Cc1ccccc1)NS(=O)(=O)c1ccc(F)cc1

nearest known ligand 0.79

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 11/20 0.79
MMP9 P14780 9/20 0.79
ADAMTS4 O75173 1/20 0.79
MMP1 P03956 2/20 0.70
MMP3 P08254 2/20 0.70
MMP13 P45452 2/20 0.70
ADAMTS5 Q9UNA0 1/20 0.70
ALDH1A1 P00352 1/20 0.70
MAPT P10636 1/20 0.70
MMP7 P09237 1/20 0.70
POLB P06746 1/20 0.66
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
L3MBTL1 Q9Y468 2/20 0.60
TP53 P04637 1/20 0.59
CTSL P07711 1/20 0.59
CTSS P25774 1/20 0.59
CTSK P43235 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5189189 1.00 MMP2 (0.79) MMP2MMP9ADAMTS4MMP1MMP3
SCHEMBL7468716 1.00 MMP2 (0.79) MMP2MMP9ADAMTS4MMP1MMP3
SCHEMBL697591 0.90 MMP2 (0.85) MMP2MMP9ADAMTS4MMP1MMP3
SCHEMBL697592 0.90 MMP2 (0.85) MMP2MMP9ADAMTS4MMP1MMP3
SCHEMBL4188026 0.90 MMP2 (0.85) MMP2MMP9ADAMTS4MMP1MMP3
SCHEMBL11951292 0.89 L3MBTL1 (0.76) MMP2MMP9ADAMTS4MMP1MMP3
SCHEMBL11950493 0.89 L3MBTL1 (0.76) MMP2MMP9ADAMTS4MMP1MMP3
SCHEMBL32691761 0.88 MMP2 (1.00) MMP2MMP9ADAMTS4MMP1MMP3
SCHEMBL1920507 0.88 MMP2 (1.00) MMP2MMP9ADAMTS4MMP1MMP3
SCHEMBL6545297 0.88 MMP2 (1.00) MMP2MMP9ADAMTS4MMP1MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0874836-B1 SULFONAMIDE INHIBITORS OF MATRIX METALLOPROTEINASES WARNER LAMBERT CO (US) 2002-10-09 EP disclosed
US-6297247-B1 Sulfonamide inhibitors of matrix metalloproteinases WARNER-LAMBERT COMPANY 2001-10-02 US disclosed
US-6153612-A Sulfonamide inhibitors of matrix metalloproteinases WARNER-LAMBERT COMPANY (US) 2000-11-28 US disclosed
US-5977141-A Sulfonamide inhibitors of matrix metalloproteinases WARNER-LAMBERT COMPANY (US) 1999-11-02 US disclosed
EP-0874836-A1 SULFONAMIDE INHIBITORS OF MATRIX METALLOPROTEINASES WARNER-LAMBERT COMPANY (US) 1998-11-04 EP disclosed
WO-1997019068-A1 SULFONAMIDE INHIBITORS OF MATRIX METALLOPROTEINASES WARNER-LAMBERT COMPANY (US) 1997-05-29 WO disclosed