SCHEMBL1920507

SCHEMBL1920507

O=C(O)[C@@H](Cc1ccccc1)NS(=O)(=O)c1ccc(-c2ccccc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 13/20 1.00
MMP9 P14780 12/20 1.00
ADAMTS4 O75173 3/20 1.00
MMP13 P45452 2/20 0.87
ADAMTS5 Q9UNA0 1/20 0.87
MMP1 P03956 1/20 0.87
MMP3 P08254 1/20 0.87
MMP7 P09237 1/20 0.87
ALDH1A1 P00352 1/20 0.73
MAPT P10636 1/20 0.73
POLB P06746 1/20 0.69
MMP8 P22894 2/20 0.68
MMP12 P39900 1/20 0.64
MMP14 P50281 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6545297 1.00 MMP2 (1.00) MMP2MMP9ADAMTS4MMP13ADAMTS5
SCHEMBL32691761 1.00 MMP2 (1.00) MMP2MMP9ADAMTS4MMP13ADAMTS5
SCHEMBL4422501 0.93 MMP2 (1.00) MMP2MMP9ADAMTS4MMP13ADAMTS5
SCHEMBL14218256 0.93 MMP2 (0.87) MMP2MMP9ADAMTS4MMP13ADAMTS5
SCHEMBL14533971 0.93 MMP2 (0.87) MMP2MMP9ADAMTS4MMP13ADAMTS5
SCHEMBL14218257 0.93 MMP2 (0.87) MMP2MMP9ADAMTS4MMP13ADAMTS5
SCHEMBL4422490 0.93 MMP2 (1.00) MMP2MMP9ADAMTS4MMP13ADAMTS5
SCHEMBL697591 0.92 MMP2 (0.85) MMP2MMP9ADAMTS4MMP13ADAMTS5
SCHEMBL4188026 0.92 MMP2 (0.85) MMP2MMP9ADAMTS4MMP13ADAMTS5
SCHEMBL697592 0.92 MMP2 (0.85) MMP2MMP9ADAMTS4MMP13ADAMTS5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 90 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100119489-A1 Stimulation of Pancreatic Beta Cell Proliferation STOFFEL MARKUS 2010-05-13 US claimed
US-20100092469-A1 ANTAGONISTS OF A NON-SELECTIVE CATION CHANNEL IN NEURAL CELLS THE U.S. OF AMERICA AS REPRESENTED BY THE DEPT OF VETERANS AFFAIRS 2010-04-15 US claimed
EP-2114160-A1 ANTAGONISTS OF A NON-SELECTIVE CATION CHANNEL IN NEURAL CELLS University of Maryland, Baltimore (US) 2009-11-11 EP claimed
WO-2008098160-A1 ANTAGONISTS OF A NON-SELECTIVE CATION CHANNEL IN NEURAL CELLS UNIVERSITY OF MARYLAND, BALTIMORE (US) 2008-08-14 WO claimed
US-12589090-B2 Compounds and methods for the treatment of degenerative disorders AQUILUS PHARMACEUTICALS, INC. (US) 2026-03-31 US disclosed
US-12121526-B2 Targeting NCCA-ATP channel for organ protection following ischemic episode THE UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS (US) 2024-10-22 US disclosed
WO-2024028417-A1 NEW COMPOSITION FOR THE TREATMENT AND/OR PREVENTION OF VITILIGO Institut National de la Santé et de la Recherche Médicale (FR) 2024-02-08 WO disclosed
US-20210113589-A1 TARGETING NCCA-ATP CHANNEL FOR ORGAN PROTECTION FOLLOWING ISCHEMIC EPISODE THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS 2021-04-22 US disclosed
US-10898496-B2 Targeting NCCa-ATP channel for organ protection following ischemic episode UNIVERSITY OF MARYLAND, BALTIMORE (US) 2021-01-26 US disclosed
WO-2020154243-A1 COMPOUNDS AND METHODS FOR THE TREATMENT OF DEGENERATIVE DISORDERS AQUILUS PHARMACEUTICALS, INC. (US) 2020-07-30 WO disclosed
US-20190117672-A1 TARGETING NCCA-ATP CHANNEL FOR ORGAN PROTECTION FOLLOWING ISCHEMIC EPISODE UNIVERSITY OF MARYLAND, BALTIMORE 2019-04-25 US disclosed
US-20190111137-A1 METHODS FOR ANTAGONISTS OF A NON-SELECTIVE CATION CHANNEL IN NEURAL CELLS UNIVERSITY OF MARYLAND, BALTIMORE 2019-04-18 US disclosed
US-20040248813-A1 Compounds and methods for the modulation of cd154 CBR INSTITUTE FOR BIOMEDICAL RESEARCH, INC. 2004-12-09 US disclosed
WO-2004105837-A2 COMPOUNDS AND METHODS FOR IMPROVING PLATELET RECOVERY AND FUNCTION CENTER FOR BLOOD RESEARCH, INC. (US) 2004-12-09 WO disclosed
US-20040205837-A1 Transgenic mouse over-expressing calreticulin (CRT) in vascular smooth muscle cells MESAELI NASRIN 2004-10-14 US disclosed
US-20040072750-A1 Compounds and methods for the modulation of CD154 MILLENNIUM PHARMACEUTICALS, INC. 2004-04-15 US disclosed
EP-1399466-A2 COMPOUNDS AND METHODS FOR THE MODULATION OF CD154 MILLENNIUM PHARMACEUTICALS, INC. (US) 2004-03-24 EP disclosed
US-20040048803-A1 Compounds and methods for the modulation of CD154 PHILLIPS DAVID (US) 2004-03-11 US disclosed
WO-2002089730-A2 COMPOUNDS AND METHODS FOR THE MODULATION OF CD154 THE CENTER FOR BLOOD RESEARCH, INC. (US) 2002-11-14 WO disclosed
US-20020165166-A1 Compounds and methods for the modulation of CD154 CBR INSTITUTE FOR BIOMEDICAL RESEARCH, INC. 2002-11-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12589090-B2 Compounds and methods for the treatment of degenerative disorders CASP3, CASP10, CASP1 MMP2 85/4885MMP9 244/4885ADAMTS4 573/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.