SCHEMBL7461012

SCHEMBL7461012

O=C=NCc1cc2ccccc2o1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.53
AGXT P21549 1/20 0.49
HTR2B P41595 2/20 0.42
HTR1A P08908 1/20 0.42
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
CYP19A1 P11511 1/20 0.41
CYP2A6 P11509 2/20 0.41
FLT3 P36888 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TYR P14679 1/20 0.40
DAO P14920 1/20 0.40
AKR1B1 P15121 1/20 0.40
HPGD P15428 1/20 0.40
POLB P06746 1/20 0.40
ADRA2A P08913 1/20 0.39
CA2 P00918 1/20 0.39
SIRT2 Q8IXJ6 2/20 0.38
SIRT1 Q96EB6 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623313 0.80 LOXL2 (0.58) LOXL2AGXTHTR2BHTR1AESR1
SCHEMBL30404454 0.80 HDAC6 (0.35) LOXL2CYP19A1FLT3POLBCA2
SCHEMBL349601 0.77 LOXL2 (0.58) LOXL2AGXTHTR2BHTR1AESR1
SCHEMBL2090461 0.74 LOXL2 (0.64) LOXL2AGXTHTR2BHTR1AESR1
SCHEMBL1259001 0.73 LOXL2 (0.54) LOXL2AGXTESR1ESR2FLT3
SCHEMBL14075637 0.73 LOXL2 (0.69) LOXL2AGXTHTR2BHTR1AESR1
SCHEMBL5541856 0.72 AGXT (0.62) LOXL2AGXTHTR2BHTR1AESR1
SCHEMBL1259643 0.72 LOXL2 (0.53) LOXL2AGXTHTR2BHTR1AESR1
SCHEMBL490975 0.71 LMNA (0.35) POLB
SCHEMBL6243293 0.71 LOXL2 (0.66) LOXL2AGXTHTR2BHTR1AESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1413206-A Non peptide tachykinin receptor antagonists WARNER LAMBERT CO (US) 2003-04-23 CN disclosed
EP-1244653-A1 NON PEPTIDE TACHYKININ RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 2002-10-02 EP disclosed
WO-2001046176-A2 NON PEPTIDE TACHYKININ RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 2001-06-28 WO disclosed