SCHEMBL7462033

SCHEMBL7462033

C#CN1CCNCC1S(=O)(=O)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 13/20 0.39
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
HTR2A P28223 2/20 0.35
HTR2C P28335 2/20 0.34
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA4 P22748 2/20 0.33
CA9 Q16790 2/20 0.33
SIGMAR1 Q99720 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30407459 0.81 CHRM2 (0.43) HTR6CHRM2CHRM1HTR2AHTR2C
SCHEMBL28061774 0.78 HTR6 (0.42) HTR6CHRM2CHRM1HTR2AHTR2C
Fluoride SCHEMBL28061775 0.77 HTR6 (0.41) HTR6CHRM2CHRM1HTR2AHTR2C
SCHEMBL3796418 0.77 SLC6A2 (0.49) HTR6CHRM2CHRM1HTR2AHTR2C
SCHEMBL6744243 0.75 CA1 (0.44) HTR6CHRM2CHRM1CTSLCTSB
SCHEMBL17004653 0.73
SCHEMBL3958698 0.73 CA1 (0.45) HTR6CHRM2CHRM1CTSLCTSB
SCHEMBL10974784 0.72 CA1 (0.39) HTR6CHRM2CHRM1HTR2AHTR2C
SCHEMBL10979646 0.72 CA1 (0.39) HTR6CHRM2CHRM1HTR2AHTR2C
SCHEMBL4552600 0.71 SIGMAR1 (0.43) HTR2AHTR2CSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0126094-A1 NEW 1,4-DIHYDROPYRIDINE ESTERS AND PREPARATION METHODS THEREOF AND DRUGS CONTAINING SAID ESTERS. CERMOL SA (CH) 1984-11-28 EP claimed
WO-1984002132-A1 NEW 1,4-DIHYDROPYRIDINE ESTERS AND PREPARATION METHODS THEREOF AND DRUGS CONTAINING SAID ESTERS CERMOL SA (CH) 1984-06-07 WO claimed
EP-0126094-B1 NEW 1,4-DIHYDROPYRIDINE ESTERS AND PREPARATION METHODS THEREOF AND DRUGS CONTAINING SAID ESTERS CERMOL S.A. (CH) 1990-06-20 EP disclosed
EP-0126094-A1 NEW 1,4-DIHYDROPYRIDINE ESTERS AND PREPARATION METHODS THEREOF AND DRUGS CONTAINING SAID ESTERS. CERMOL SA (CH) 1984-11-28 EP disclosed
WO-1984002132-A1 NEW 1,4-DIHYDROPYRIDINE ESTERS AND PREPARATION METHODS THEREOF AND DRUGS CONTAINING SAID ESTERS CERMOL SA (CH) 1984-06-07 WO disclosed