SCHEMBL7463145

SCHEMBL7463145

[CH2]c1ccc(-n2ncnn2)cc1

nearest known ligand 0.35

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 1/20 0.35
PDPK1 O15530 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7400517 0.77 CYP2A6 (0.36) BRS3PDPK1
SCHEMBL9440546 0.77 NOTUM (0.45) BRS3
Hydrochloric Acid SCHEMBL4739527 0.76 NOTUM (0.44) BRS3
SCHEMBL8470236 0.75 PDPK1 (0.35) PDPK1
SCHEMBL14895448 0.71 ALDH1A1 (0.40) BRS3PDPK1
SCHEMBL7402637 0.67 ADH5 (0.47)
SCHEMBL7321916 0.65 KDM4E (0.46) PDPK1
SCHEMBL16897456 0.64 CXCR2 (0.36) BRS3
SCHEMBL676377 0.62 SMN1; SMN2 (0.60) BRS3
SCHEMBL4582384 0.62 NOTUM (0.64)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1021181-A4 CARBOXYLIC ACID INDOLE INHIBITORS OF CHEMOKINES SMITHKLINE BEECHAM CORP (US) 2002-06-26 EP disclosed
EP-1021181-A1 CARBOXYLIC ACID INDOLE INHIBITORS OF CHEMOKINES SMITHKLINE BEECHAM CORPORATION (US) 2000-07-26 EP disclosed
US-5955492-A Carboxylic acid indole inhibitors of chemokines SMITHKLINE BEECHAM CORPORATION (US) 1999-09-21 US disclosed
WO-1997035572-A1 CARBOXYLIC ACID INDOLE INHIBITORS OF CHEMOKINES SMITHKLINE BEECHAM CORPORATION (US) 1997-10-02 WO disclosed