SCHEMBL7463397

SCHEMBL7463397

C=CCn1c(C(F)(F)F)cc(=O)n(-c2ccc3snc(-c4cc(OCC(=O)O)ccc4C)c3c2)c1=O

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.34
ADORA2B P29275 2/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA1 P30542 1/20 0.34
PPARD Q03181 13/20 0.33
AGER Q15109 1/20 0.32
NR4A1 P22736 1/20 0.31
APEX1 P27695 1/20 0.31
BLK P51451 1/20 0.31
BMX P51813 1/20 0.31
JAK3 P52333 1/20 0.31
BTK Q06187 1/20 0.31
MEN1 O00255 1/20 0.30
POLB P06746 1/20 0.30
KMT2A Q03164 1/20 0.30
PPARA Q07869 2/20 0.30
SYK P43405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7468473 0.91 FABP4 (0.35) ADORA2AADORA2BPPARDAGERNR4A1
SCHEMBL7459571 0.88 AGER (0.35) ADORA2BPPARDAGERNR4A1APEX1
SCHEMBL7463386 0.87 PTGDR2 (0.35) PPARDPPARA
SCHEMBL7467248 0.83 TP53 (0.32) ADORA2AADORA2BAGERPOLB
SCHEMBL7454798 0.82 PPARD (0.35) PPARDAGERNR4A1APEX1MEN1
SCHEMBL7468039 0.81 KDM4E (0.39) ADORA2AADORA2BPPARDNR4A1APEX1
SCHEMBL7458882 0.80 POLB (0.41) PPARDAGERNR4A1APEX1MEN1
SCHEMBL7459459 0.80 LMNA (0.32) KMT2A
SCHEMBL7461737 0.79 ALPL (0.37) PPARDAGERNR4A1APEX1POLB
SCHEMBL8087543 0.79

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0908457-B1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents BASF AG (DE) 2002-11-13 EP disclosed
EP-0908457-A1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents American Cyanamid Company (US) 1999-04-14 EP disclosed