SCHEMBL7463510

SCHEMBL7463510

CN1CC(C(=O)N(CCCN2CCN(c3ccc(F)cc3)CC2)c2ccccc2)CC1=O

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 2/20 0.48
HTR1A P08908 3/20 0.47
HTR7 P34969 3/20 0.46
HTR2A P28223 3/20 0.46
HTR2C P28335 3/20 0.46
DRD2 P14416 4/20 0.45
DRD4 P21917 4/20 0.45
DRD3 P35462 3/20 0.45
HRH1 P35367 1/20 0.45
TP53 P04637 1/20 0.44
CYP1A2 P05177 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7469296 0.97 HTR1A (0.47) CCR5HTR1AHTR7HTR2AHTR2C
SCHEMBL5073448 0.85 KDM4E (0.56) CCR5HTR2AHTR2CCYP1A2
Hydrochloric Acid SCHEMBL7465744 0.84 CCR5 (0.62) CCR5
SCHEMBL7464238 0.84 CCR5 (0.53) CCR5
Hydrochloric Acid SCHEMBL7468181 0.83 CCR5 (0.50) CCR5HTR2ADRD3
SCHEMBL7458312 0.83 KDM4E (0.58) CCR5HTR2AHTR2CCYP1A2
Hydrochloric Acid SCHEMBL7470069 0.83 CCR5 (0.52) CCR5
SCHEMBL7455494 0.82 CCR5 (0.49) CCR5DRD3
SCHEMBL7464185 0.82 KDM4E (0.57) CCR5HTR2AHTR2CCYP1A2
SCHEMBL7456202 0.82 CCR5 (0.49) CCR5HTR2ADRD2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1180513-A1 CYCLIC AMIDE COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-02-20 EP disclosed