SCHEMBL7464185

SCHEMBL7464185

CN1CC(C(=O)N(CCCCCN2CCC(C(=O)c3ccc(F)cc3)CC2)c2ccccc2)CC1=O

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.57
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
HTR2A P28223 1/20 0.57
KCNH2 Q12809 2/20 0.49
CCR5 P51681 1/20 0.47
HTR2C P28335 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7458312 0.99 KDM4E (0.58) KDM4ECYP1A2CYP3A4CYP2D6HTR2A
SCHEMBL5073448 0.96 KDM4E (0.56) KDM4ECYP1A2CYP3A4CYP2D6HTR2A
Fumaric Acid SCHEMBL7464795 0.90 HTR2A (0.50) KDM4ECYP1A2CYP3A4CYP2D6HTR2A
Fumaric Acid SCHEMBL7464788 0.90 HTR2A (0.50) KDM4ECYP1A2CYP3A4CYP2D6HTR2A
SCHEMBL7469296 0.85 HTR1A (0.47) HTR2ACCR5HTR2C
SCHEMBL7464796 0.84 HTR2A (0.48) KDM4ECYP1A2CYP3A4CYP2D6HTR2A
Hydrochloric Acid SCHEMBL7458703 0.84 CCR5 (0.59) KCNH2CCR5
Hydrochloric Acid SCHEMBL7465744 0.83 CCR5 (0.62) CCR5
SCHEMBL7463510 0.82 CCR5 (0.48) CYP1A2HTR2ACCR5HTR2C
Hydrochloric Acid SCHEMBL7468181 0.79 CCR5 (0.50) CYP2D6HTR2ACCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1180513-A1 CYCLIC AMIDE COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-02-20 EP disclosed