SCHEMBL7464796

SCHEMBL7464796

CN1CC(C(=O)N(CC(O)CN2CCC(C(=O)c3ccc(F)cc3)CC2)c2ccccc2)CC1=O

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.48
KDM4E B2RXH2 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
ADRB2 P07550 1/20 0.44
ADRB1 P08588 1/20 0.44
ADRB3 P13945 1/20 0.44
HTR2C P28335 2/20 0.44
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HTR7 P34969 1/20 0.43
HTR6 P50406 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5073448 0.86 KDM4E (0.56) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL7458312 0.85 KDM4E (0.58) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
Fumaric Acid SCHEMBL7464795 0.84 HTR2A (0.50) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL7464185 0.84 KDM4E (0.57) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
Fumaric Acid SCHEMBL7464788 0.84 HTR2A (0.50) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL7458703 0.74 CCR5 (0.59)
Hydrochloric Acid SCHEMBL7465744 0.72 CCR5 (0.62)
SCHEMBL7463510 0.71 CCR5 (0.48) HTR2ACYP1A2HTR2CHTR7
SCHEMBL7469296 0.71 HTR1A (0.47) HTR2AHTR2CHTR7
SCHEMBL10722200 0.71 HTR2A (0.59) HTR2AKDM4ECYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1180513-A1 CYCLIC AMIDE COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-02-20 EP disclosed