SCHEMBL7464316

SCHEMBL7464316

c1ccc(COc2ccccc2-c2ncccn2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.59
LTA4H P09960 1/20 0.59
MAPK14 Q16539 1/20 0.59
ADRA1A P35348 1/20 0.56
SGMS2 Q8NHU3 1/20 0.55
PDE5A O76074 1/20 0.55
PDE4A P27815 1/20 0.55
PDE4B Q07343 1/20 0.55
PDE4C Q08493 1/20 0.55
PDE4D Q08499 1/20 0.55
IDO1 P14902 1/20 0.54
MAPT P10636 1/20 0.52
MAPK1 P28482 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
RXRA P19793 1/20 0.51
RXRB P28702 1/20 0.51
RXRG P48443 1/20 0.51
PTGER1 P34995 3/20 0.51
ABCB1 P08183 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7462666 0.89 LTA4H (0.51) BRD4LTA4HMAPK14ADRA1ASGMS2
SCHEMBL26013299 0.84 MAPT (0.63) BRD4LTA4HMAPK14SGMS2IDO1
SCHEMBL8210963 0.82 BRD4 (0.53) BRD4LTA4HMAPK14ADRA1ASGMS2
SCHEMBL28284772 0.82 ADRA1D (0.58) BRD4LTA4HMAPK14ADRA1ASGMS2
SCHEMBL9566443 0.80 BRD4 (0.57) BRD4LTA4HMAPK14SGMS2PDE5A
SCHEMBL1423699 0.79 CYP11B1 (0.60) BRD4LTA4HMAPK14ADRA1ASGMS2
SCHEMBL201074 0.79 RXRA (0.70) BRD4ADRA1AIDO1MAPTMAPK1
SCHEMBL16416752 0.78 LTA4H (0.64) LTA4HMAPK14SGMS2PDE5APDE4A
SCHEMBL339812 0.77 MAPT (0.71) BRD4LTA4HMAPK14ADRA1AIDO1
SCHEMBL28185277 0.77 PDE5A (0.53) ADRA1APDE5AMAPTTDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0817773-B1 PYRIMIDINE COMPOUNDS QINETIQ LTD (GB) 2002-06-12 EP disclosed
US-6121448-A LIQUID CRYSTALLINE COMPOUNDS THE SECRETARY OF STATE FOR DEFENCE IN HER BRITTANIC MAJESTY'S GOVERNMENT OF THE UNITED KINGDOM OF GREAT BRITAIN AND NORTHERN IRELAND (GB) 2000-09-19 US disclosed
US-5986096-A REACTION OF HYDROGEN IODIDE WITH CHLORO-5-BROMOPYRIMIDINE THE SECRETARY OF STATE FOR DEFENCE IN HER BRITANNIC MAJESTY'S A GOVERNMENT OF THE U.K. OF GT. BRITAIN & N. IRELAND OF DEFENCE EVALUATION & RESEARCH AGENCY (GB) 1999-11-16 US disclosed
WO-1996030344-A9 PYRIMIDINE COMPOUNDS 1999-02-11 WO disclosed
WO-1996030344-A2 PYRIMIDINE COMPOUNDS THE SECRETARY OF STATE FOR DEFENCE (GB) 1996-10-03 WO disclosed