SCHEMBL7464319

SCHEMBL7464319

c1ccc(COc2ccnc(-c3ccccc3)n2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.50
ALKBH1 Q13686 1/20 0.48
CLK4 Q9HAZ1 3/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 2/20 0.42
MAPT P10636 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
XDH P47989 1/20 0.41
CYP3A4 P08684 4/20 0.41
CYP1A2 P05177 3/20 0.41
CYP2D6 P10635 3/20 0.41
CYP2C19 P33261 3/20 0.41
USP2 O75604 1/20 0.41
GABRA5 P31644 2/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA3 P34903 1/20 0.40
ALDH1A1 P00352 2/20 0.40
TP53 P04637 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29111010 0.85 ALKBH1 (0.41) PDE5AALKBH1CLK4MEN1KMT2A
SCHEMBL23767729 0.84 ALKBH1 (0.51) ALKBH1MEN1KMT2AXDHCYP3A4
SCHEMBL1163902 0.84 XDH (0.45) PDE5AALKBH1CLK4MEN1KMT2A
SCHEMBL30080246 0.84 ALKBH1 (0.51) ALKBH1MEN1KMT2AXDHCYP3A4
SCHEMBL25544486 0.82 ALKBH1 (0.49) ALKBH1CLK4MEN1KMT2AXDH
SCHEMBL30080394 0.82 ALKBH1 (0.49) ALKBH1MEN1KMT2AL3MBTL1XDH
SCHEMBL23767730 0.82 ALKBH1 (0.49) ALKBH1MEN1KMT2AL3MBTL1XDH
SCHEMBL23753904 0.81 SMN1; SMN2 (0.54) ALKBH1CLK4MEN1KMT2AMAPT
SCHEMBL13763835 0.81 ALDH1A1 (0.47) CLK4MEN1KMT2AKDM4EMAPT
SCHEMBL23767728 0.80 ALKBH1 (0.47) ALKBH1CLK4KDM4EL3MBTL1XDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0817773-B1 PYRIMIDINE COMPOUNDS QINETIQ LTD (GB) 2002-06-12 EP disclosed
US-6121448-A LIQUID CRYSTALLINE COMPOUNDS THE SECRETARY OF STATE FOR DEFENCE IN HER BRITTANIC MAJESTY'S GOVERNMENT OF THE UNITED KINGDOM OF GREAT BRITAIN AND NORTHERN IRELAND (GB) 2000-09-19 US disclosed
US-5986096-A REACTION OF HYDROGEN IODIDE WITH CHLORO-5-BROMOPYRIMIDINE THE SECRETARY OF STATE FOR DEFENCE IN HER BRITANNIC MAJESTY'S A GOVERNMENT OF THE U.K. OF GT. BRITAIN & N. IRELAND OF DEFENCE EVALUATION & RESEARCH AGENCY (GB) 1999-11-16 US disclosed
WO-1996030344-A9 PYRIMIDINE COMPOUNDS 1999-02-11 WO disclosed
WO-1996030344-A2 PYRIMIDINE COMPOUNDS THE SECRETARY OF STATE FOR DEFENCE (GB) 1996-10-03 WO disclosed