SCHEMBL7464415

SCHEMBL7464415

[CH2]C(CCCCCC)c1c(Cl)cccc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KCNH2 Q12809 2/20 0.35
CSNK1E P49674 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
EPHX2 P34913 1/20 0.34
OPRM1 P35372 4/20 0.34
OPRD1 P41143 4/20 0.34
OPRK1 P41145 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7471569 0.81 KDM4E (0.39) MEN1KMT2ASMN1; SMN2KDM4ELMNA
SCHEMBL20178499 0.80 MEN1 (0.43) MEN1KMT2ATP53CYP1A2CYP3A4
SCHEMBL18567612 0.78 MEN1 (0.40) MEN1KMT2ATP53CYP1A2CYP3A4
SCHEMBL4428343 0.77 MEN1 (0.40) MEN1KMT2ATP53CYP1A2CYP3A4
SCHEMBL7470789 0.76 OPRM1 (0.48) EPHX2OPRM1OPRD1OPRK1OPRL1
SCHEMBL28058440 0.74 OPRM1 (0.47) KMT2AEPHX2OPRM1OPRD1OPRK1
SCHEMBL16951539 0.74 PNMT (0.46) MEN1KMT2ACYP1A2CYP3A4TSHR
SCHEMBL24950078 0.73 NR1I2 (0.39) MEN1KMT2ATP53CYP1A2CYP3A4
SCHEMBL15351833 0.73 SLC6A2 (0.44) SMN1; SMN2KDM4EKCNH2SLC6A4SLC6A3
SCHEMBL23101932 0.72 MEN1 (0.47) MEN1KMT2ATP53CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244617-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE Ortho-McNeil Pharmaceutical, Inc. (US) 2002-10-02 EP disclosed
WO-2001047875-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-07-05 WO disclosed