SCHEMBL7464639

SCHEMBL7464639

COc1ccc2nc3c(c(Cl)c2c1)C(=O)c1ccccc1-3

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.60
ADORA2A P29274 2/20 0.50
ADORA1 P30542 2/20 0.50
C1R P00736 1/20 0.46
ACHE P22303 4/20 0.46
BCHE P06276 2/20 0.46
PDE4B Q07343 2/20 0.46
PDE4D Q08499 2/20 0.46
L3MBTL1 Q9Y468 3/20 0.45
PPARG P37231 1/20 0.45
HTT P42858 1/20 0.45
NCOA2 Q15596 1/20 0.45
NCOA1 Q15788 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
NCOA3 Q9Y6Q9 1/20 0.45
MAPT P10636 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
PKM P14618 2/20 0.43
MAPK1 P28482 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7458826 0.90 TP53 (0.60) TP53ADORA2AADORA1ACHEBCHE
SCHEMBL7464351 0.86 ACHE (0.51) TP53ADORA2AADORA1ACHEPDE4B
SCHEMBL7464693 0.86 ACHE (0.51) TP53ADORA2AADORA1ACHEPDE4B
SCHEMBL7820175 0.81 TP53 (0.51) TP53ADORA2AADORA1C1RACHE
SCHEMBL7464904 0.80 ESRRB (0.45) TP53ADORA2AADORA1HTTRXFP1
SCHEMBL12285138 0.74 KDM4E (0.55) ACHEBCHESMN1; SMN2NPC1RAB9A
SCHEMBL13739299 0.73 KMT2A (0.61) L3MBTL1HTTMAPTSMN1; SMN2NPC1
SCHEMBL7825423 0.73 TP53 (0.51) TP53ADORA2AADORA1PDE4BPDE4D
SCHEMBL7533761 0.72 KDM4E (0.54) MAPTSMN1; SMN2NPC1MAOBRAB9A
SCHEMBL7811355 0.72 NTRK1 (0.50) TP53ACHEPDE4BPDE4DKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785191-B1 FUSED INDAN DERIVATIVES AND SALTS THEREOF TAIHO PHARMACEUTICAL CO LTD (JP) 2002-10-23 EP disclosed
US-5763453-A ANTITUMOR AGENTS TAIHO PHARMACEUTICAL CO., LTD. (JP) 1998-06-09 US disclosed
EP-0785191-A1 FUSED INDAN DERIVATIVES AND SALTS THEREOF TAIHO PHARMACEUTICAL CO., LTD. (JP) 1997-07-23 EP disclosed