SCHEMBL7464863

SCHEMBL7464863

FC(F)(F)c1ccccc1C(Oc1[c]cccc1)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 6/20 0.45
TDO2 P48775 6/20 0.45
ACP3 P15309 1/20 0.41
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
OPRL1 P41146 1/20 0.34
CACNA2D1 P54289 1/20 0.33
CACNA1B Q00975 1/20 0.33
CACNB1 Q02641 1/20 0.33
CACNA1C Q13936 1/20 0.33
CNR2 P34972 1/20 0.33
SLC6A4 P31645 1/20 0.30
IDO2 Q6ZQW0 1/20 0.30
PPARG P37231 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7460305 0.81 IDO1 (0.53) IDO1TDO2OPRM1OPRD1OPRK1
SCHEMBL7471840 0.79 ACP3 (0.42) IDO1TDO2ACP3OPRM1OPRK1
SCHEMBL7471512 0.79 SRD5A2 (0.36) IDO1TDO2OPRM1OPRK1SLC6A4
SCHEMBL7458608 0.78 ESR1 (0.46) IDO1TDO2ACP3OPRM1SLC6A4
SCHEMBL7456441 0.77 IDO1 (0.54) IDO1TDO2OPRM1OPRD1OPRK1
SCHEMBL11343236 0.76 IDO1 (0.55) IDO1TDO2ACP3OPRM1OPRD1
SCHEMBL7465983 0.76 IDO1 (0.57) IDO1TDO2ACP3OPRM1OPRD1
SCHEMBL7470957 0.75 IDO1 (0.43) IDO1TDO2ACP3OPRM1OPRD1
SCHEMBL7466004 0.74 IDO1 (0.40) IDO1TDO2SLC6A4
SCHEMBL7466815 0.71 MEN1 (0.37) IDO1TDO2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244617-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE Ortho-McNeil Pharmaceutical, Inc. (US) 2002-10-02 EP claimed
WO-2001047875-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-07-05 WO claimed