SCHEMBL7465152

SCHEMBL7465152

Oc1cnc(-c2cccc(F)c2F)nc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.40
BCAT1 P54687 1/20 0.38
CES2 O00748 1/20 0.35
BCHE P06276 1/20 0.35
CES1 P23141 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
GRM5 P41594 2/20 0.35
PTPN11 Q06124 1/20 0.35
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
CCNE2 O96020 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
CYP11B1 P15538 2/20 0.33
HSD11B1 P28845 1/20 0.33
WDR5 P61964 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6270187 0.79 CCNE2 (0.41) CNR2BCAT1CES2BCHECES1
SCHEMBL3038641 0.71 CES2 (0.46) CNR2BCAT1CES2BCHECES1
SCHEMBL1513514 0.69 ABL1 (0.47) CNR2CES2BCHECES1HDAC3
SCHEMBL11907633 0.69 ATR (0.38) CNR2HDAC6GRM5GSK3AGSK3B
SCHEMBL14832981 0.69 ALB (0.43) BCAT1CES2BCHECES1WDR5
SCHEMBL9276928 0.68 ESR2 (0.48) CNR2HDAC3HDAC1HDAC2HDAC8
SCHEMBL23251236 0.68 ALDH1A1 (0.47) NPC1
SCHEMBL27341090 0.67 MAOA (0.46) BCAT1CES2BCHECES1CDK2
SCHEMBL6367917 0.67 ALDH1A1 (0.44) CES2BCHECES1PIK3CANPC1
SCHEMBL5189298 0.67 CNR2 (0.51) CNR2BCAT1HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0817773-B1 PYRIMIDINE COMPOUNDS QINETIQ LTD (GB) 2002-06-12 EP disclosed
US-6121448-A LIQUID CRYSTALLINE COMPOUNDS THE SECRETARY OF STATE FOR DEFENCE IN HER BRITTANIC MAJESTY'S GOVERNMENT OF THE UNITED KINGDOM OF GREAT BRITAIN AND NORTHERN IRELAND (GB) 2000-09-19 US disclosed
US-5986096-A REACTION OF HYDROGEN IODIDE WITH CHLORO-5-BROMOPYRIMIDINE THE SECRETARY OF STATE FOR DEFENCE IN HER BRITANNIC MAJESTY'S A GOVERNMENT OF THE U.K. OF GT. BRITAIN & N. IRELAND OF DEFENCE EVALUATION & RESEARCH AGENCY (GB) 1999-11-16 US disclosed
WO-1996030344-A9 PYRIMIDINE COMPOUNDS 1999-02-11 WO disclosed