SCHEMBL7465981

SCHEMBL7465981

CCOC(=O)CCNC(=O)CN1CCN(c2ccc3c(c2)CCN(C(=O)OC(C)(C)C)CC3)C1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.40
ESR2 Q92731 1/20 0.39
TMEM97 Q5BJF2 2/20 0.38
SIGMAR1 Q99720 2/20 0.38
HTR1A P08908 1/20 0.38
CHRM5 P08912 1/20 0.38
SLC6A2 P23975 1/20 0.38
HRH2 P25021 1/20 0.38
ADRA1D P25100 1/20 0.38
HTR1B P28222 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR1E P28566 1/20 0.38
HRH1 P35367 1/20 0.38
HTR2B P41595 1/20 0.38
SLC6A3 Q01959 1/20 0.38
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
ITGB3 P05106 2/20 0.36
ITGA2B P08514 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7481405 0.82 NR1H2 (0.42) NR1H2ESR2NPC1RAB9AITGB3
SCHEMBL7468291 0.82 NR1H2 (0.38) NR1H2ESR2TMEM97SIGMAR1HTR1A
SCHEMBL7419930 0.81 NR1H2 (0.49) NR1H2ESR2TMEM97SIGMAR1NPC1
SCHEMBL7479149 0.81 ITGB3 (0.40) TMEM97SIGMAR1HTR1ACHRM5SLC6A2
SCHEMBL7381195 0.80 ITGB3 (0.56) TMEM97SIGMAR1HTR1ACHRM5SLC6A2
SCHEMBL7474864 0.78 TMEM97 (0.39) NR1H2ESR2TMEM97SIGMAR1HTR1A
SCHEMBL7473247 0.78 NR1H2 (0.47) NR1H2ESR2TMEM97SIGMAR1NPC1
SCHEMBL7474006 0.77 ITGB3 (0.38) TMEM97SIGMAR1HTR1ACHRM5SLC6A2
SCHEMBL7468971 0.76 ITGB3 (0.42) NR1H2ESR2NPC1RAB9AITGB3
SCHEMBL7474275 0.76 ITGB3 (0.51) RAB9AITGB3ITGA2BKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777667-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT Dr. Karl Thomae GmbH (DE) 1997-06-11 EP disclosed
WO-1996005194-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT DR. KARL THOMAE GMBH (DE) 1996-02-22 WO disclosed