SCHEMBL7419930

SCHEMBL7419930

CC(C)(C)OC(=O)N1CCc2ccc(N3CCN(CC(=O)O)C3=O)cc2CC1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.49
ESR2 Q92731 2/20 0.47
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
USP30 Q70CQ3 2/20 0.39
GPR119 Q8TDV5 6/20 0.38
MAPT P10636 3/20 0.37
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
THRB P10828 1/20 0.37
LMNA P02545 1/20 0.37
EP300 Q09472 1/20 0.36
HDAC1 Q13547 1/20 0.36
TMEM97 Q5BJF2 2/20 0.36
SIGMAR1 Q99720 2/20 0.36
JAK2 O60674 2/20 0.36
JAK3 P52333 2/20 0.36
PTK2 Q05397 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7473247 0.90 NR1H2 (0.47) NR1H2ESR2NPC1RAB9AUSP30
SCHEMBL7468971 0.84 ITGB3 (0.42) NR1H2ESR2NPC1RAB9AUSP30
SCHEMBL7481405 0.83 NR1H2 (0.42) NR1H2ESR2NPC1RAB9AGPR119
Hydrochloric Acid SCHEMBL7472463 0.82 DRD3 (0.42) MAPTALDH1A1KDM4ELMNAEP300
SCHEMBL7465981 0.81 NR1H2 (0.40) NR1H2ESR2NPC1RAB9AGPR119
SCHEMBL20929267 0.78 NR1H2 (0.64) NR1H2ESR2NPC1RAB9AUSP30
SCHEMBL8565729 0.77 NR1H2 (0.45) NR1H2ESR2NPC1RAB9AUSP30
SCHEMBL7478863 0.77 NR1H2 (0.54) NR1H2ESR2NPC1RAB9AUSP30
SCHEMBL7477263 0.77 USP30 (0.51) NR1H2ESR2NPC1RAB9AUSP30
SCHEMBL7468291 0.76 NR1H2 (0.38) NR1H2ESR2NPC1RAB9AGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777667-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT Dr. Karl Thomae GmbH (DE) 1997-06-11 EP disclosed
WO-1996005194-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT DR. KARL THOMAE GMBH (DE) 1996-02-22 WO disclosed