SCHEMBL7466186

SCHEMBL7466186

CC(=O)Nc1ccc(OP(=O)(CN[C@@H](Cc2ccc(-c3ccccc3)cc2)C(=O)O)Oc2ccc(NC(C)=O)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 2/20 0.47
NPR3 P17342 1/20 0.46
F2 P00734 2/20 0.44
F10 P00742 2/20 0.44
PLG P00747 2/20 0.44
PLAU P00749 2/20 0.44
PLAT P00750 2/20 0.44
PPARG P37231 6/20 0.43
PPARA Q07869 5/20 0.43
PTGIR P43119 2/20 0.42
CYP2C9 P11712 1/20 0.42
PTGER4 P35408 1/20 0.42
PTGER2 P43116 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
MME P08473 1/20 0.42
ACE P12821 1/20 0.42
CPA1 P15085 1/20 0.42
ACE2 Q9BYF1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7410891 0.91 FPR2 (0.46) FPR2NPR3F2F10PLG
SCHEMBL7407175 0.88 MME (0.48) PPARGPPARAMMEACECPA1
SCHEMBL7318259 0.86 MMEL1 (0.49)
SCHEMBL31510352 0.81 ANPEP (0.48) FPR2L3MBTL1MEN1KMT2AMME
SCHEMBL7412181 0.81 MME (0.44) PPARGPPARAMEN1KMT2AMME
SCHEMBL8923752 0.81 MME (0.43) NPR3F2F10PLGPLAU
SCHEMBL7419794 0.81 MME (0.50) MEN1KMT2AMME
SCHEMBL7315613 0.80 HDAC8 (0.44) CYP2C9MEN1KMT2A
SCHEMBL7413775 0.80 PPARG (0.49) PPARGPPARAMMEACECPA1
SCHEMBL7415659 0.80 KMT2A (0.48) FPR2KMT2AMMEACECPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0660840-B1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES CIBA GEIGY AG (CH) 1997-05-07 EP disclosed
WO-1996026729-A1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES AS ECE INHIBITORS CIBA-GEIGY AG (CH) 1996-09-06 WO disclosed
US-5550119-A ENDOTHELIN-CONVERTING ENZYM INHIBITORS CIBA-GEIGY CORPORATION (US) 1996-08-27 US disclosed
EP-0660840-A1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES. CIBA GEIGY AG (CH) 1995-07-05 EP disclosed
WO-1994005677-A1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1994-03-17 WO disclosed
US-5250522-A Neutral endopeptidase inhibitors; cardiovascular disorders CIBA-GEIGY CORPORATION (US) 1993-10-05 US disclosed