SCHEMBL7466847

SCHEMBL7466847

Nc1ncc(-c2ccc(-n3ccnc3)cc2)c(-c2cccnc2)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 6/20 0.50
ADORA2A P29274 4/20 0.50
CYP3A4 P08684 5/20 0.49
TSHR P16473 3/20 0.49
CYP1A2 P05177 3/20 0.49
TDP1 Q9NUW8 2/20 0.49
ALOX15 P16050 2/20 0.49
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.49
CYP2A6 P11509 1/20 0.47
ACVR1 Q04771 1/20 0.46
CYP2D6 P10635 3/20 0.46
LMNA P02545 2/20 0.46
HSD17B10 Q99714 2/20 0.46
ALDH1A1 P00352 1/20 0.46
MAPK1 P28482 1/20 0.46
MAPT P10636 1/20 0.44
ABL1 P00519 1/20 0.43
PDGFRB P09619 1/20 0.43
BCR P11274 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7471062 0.88 ABL1 (0.51) ADORA1ADORA2ACYP3A4TSHRCYP1A2
SCHEMBL7462501 0.86 ADORA1 (0.60) ADORA1ADORA2ACYP3A4TSHRALOX15
SCHEMBL7535967 0.82 MEN1 (0.48) ADORA1ADORA2ACYP3A4TSHRCYP1A2
SCHEMBL6832429 0.81 ADORA1 (0.61) ADORA1ADORA2AKMT2AHSP90AA1HSP90AB1
SCHEMBL28118705 0.80 ADORA1 (0.74) ADORA1ADORA2AKMT2AHSP90AA1HSP90AB1
SCHEMBL7463419 0.78 ADORA1 (0.59) ADORA1ADORA2AABL1PDGFRBBCR
SCHEMBL6831577 0.73 MEN1 (0.59) ADORA1ADORA2AMEN1MKNK1MKNK2
SCHEMBL7468146 0.73 DHFR (0.48) ADORA1ADORA2AABL1PDGFRBBCR
SCHEMBL6832217 0.72 ADORA1 (0.53) ADORA1ADORA2AKMT2ACYP2A6HSP90AA1
SCHEMBL7467735 0.71 ADORA1 (0.42) ADORA1ADORA2ALMNAALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233461-B2 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 2002-05-29 EP disclosed