SCHEMBL7466905

SCHEMBL7466905

NC(=O)C(CO)NCCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.45
SIGMAR1 Q99720 2/20 0.45
ALDH1A1 P00352 2/20 0.45
LMNA P02545 2/20 0.45
CA12 O43570 2/20 0.45
CA2 P00918 2/20 0.45
CA9 Q16790 2/20 0.45
KDM4E B2RXH2 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
BLM P54132 1/20 0.45
GFER P55789 1/20 0.45
PMP22 Q01453 1/20 0.45
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
GGT1 P19440 1/20 0.44
NPC1 O15118 1/20 0.44
KDM1A O60341 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8054827 1.00 CYP3A4 (0.45) CYP3A4SIGMAR1ALDH1A1LMNACA12
SCHEMBL7466897 1.00 CYP3A4 (0.45) CYP3A4SIGMAR1ALDH1A1LMNACA12
SCHEMBL8211584 0.90 GGT1 (0.56) SIGMAR1LMNAKDM4EGAACYP2D6
SCHEMBL8211581 0.90 GGT1 (0.56) SIGMAR1LMNAKDM4EGAACYP2D6
Hydrochloric Acid SCHEMBL8209005 0.89 GGT1 (0.55) SIGMAR1KDM4EGAACYP2D6CYP2C9
Hydrochloric Acid SCHEMBL8209008 0.89 GGT1 (0.55) SIGMAR1KDM4EGAACYP2D6CYP2C9
Hydrochloric Acid SCHEMBL11100782 0.89 GGT1 (0.55) SIGMAR1KDM4EGAACYP2D6CYP2C9
SCHEMBL30882505 0.87 OPRK1 (0.49) CYP3A4SIGMAR1ALDH1A1LMNACA12
SCHEMBL30882671 0.87 OPRK1 (0.49) CYP3A4SIGMAR1ALDH1A1LMNACA12
SCHEMBL7469306 0.86 GGT1 (0.54) CYP3A4SIGMAR1ALDH1A1LMNACA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0764648-B1 Cephem derivatives and process for the preparation thereof EISAI CO LTD (JP) 2002-01-16 EP disclosed
EP-0333154-B1 Process for the preparation of cephem derivatives EISAI CO LTD (JP) 1997-07-16 EP disclosed
EP-0764648-A1 Cephem derivatives and process for the preparation thereof Eisai Co., Ltd. (JP) 1997-03-26 EP disclosed
EP-0612751-A2 Compounds for the preparation of cephem derivatives Eisai Co., Ltd. (JP) 1994-08-31 EP disclosed
US-5128465-A Containing thiadiazole ring and fluorine substitution EISAI CO., LTD. (JP) 1992-07-07 US disclosed
EP-0333154-A2 Process for the preparation of cephem derivatives and intermediates therefor Eisai Co., Ltd. (JP) 1989-09-20 EP disclosed