SCHEMBL7466958

SCHEMBL7466958

CSc1ccc(-c2cc(C(F)F)nn2-c2ccc(C(C)=O)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.55
PTGS1 P23219 10/20 0.50
ALDH1A1 P00352 2/20 0.42
ABCB11 O95342 1/20 0.42
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7456119 0.91 PTGS2 (0.67) PTGS2PTGS1ALDH1A1ABCB11HPGD
SCHEMBL7465548 0.90 PTGS2 (0.54) PTGS2PTGS1ALDH1A1ABCB11HDAC3
SCHEMBL8924204 0.90 PTGS2 (0.57) PTGS2PTGS1ALDH1A1ABCB11HPGD
SCHEMBL5149168 0.85 PTGS2 (0.51) PTGS2PTGS1ALDH1A1ABCB11
SCHEMBL9210879 0.84 PTGS2 (0.62) PTGS2PTGS1ALDH1A1ABCB11
SCHEMBL8638291 0.83 ALDH1A1 (0.56) PTGS2PTGS1ALDH1A1HDAC3HDAC4
SCHEMBL9206762 0.83 PTGS2 (0.54) PTGS2PTGS1ALDH1A1ABCB11
SCHEMBL7465558 0.83 PTGS2 (0.66) PTGS2PTGS1
SCHEMBL8639953 0.82 PTGS2 (0.48) PTGS2PTGS1ALDH1A1ABCB11
SCHEMBL8953830 0.81 PTGS2 (0.61) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0554829-B1 Pyrazole derivatives with antiinflammatory, analgesic and antithrombolic activity FUJISAWA PHARMACEUTICAL CO (JP) 2002-05-15 EP disclosed
EP-0856000-A1 1,3,5-TRISUBSTITUTED PYRAZOLES FOR TREAMENT OF INFLAMMATION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-08-05 EP disclosed
US-5670533-A ANTIINFLAMMATORY AGENTS, ANALGESICS OR ANTIRHEUMATIC DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-09-23 US disclosed
WO-1997013755-A1 1,3,5-TRISUBSTITUTED PYRAZOLES FOR TREAMENT OF INFLAMMATION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-04-17 WO disclosed
US-5550147-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTITHROMBOTIC AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-08-27 US disclosed
EP-0554829-A2 Pyrazole derivatives with antiinflammatory, analgesic and antithrombolic activity FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-08-11 EP disclosed