SCHEMBL8638291

SCHEMBL8638291

CSc1ccc(-c2cc(C)nn2-c2ccc(C(C)=O)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.56
HPGD P15428 3/20 0.56
CYP1A2 P05177 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
RECQL P46063 1/20 0.54
MAPT P10636 3/20 0.52
PTGS2 P35354 5/20 0.52
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
PTGS1 P23219 1/20 0.46
ALOX5 P09917 1/20 0.45
USP2 O75604 1/20 0.45
MAPK1 P28482 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.42
KDM5A P29375 1/20 0.42
KDM4C Q9H3R0 1/20 0.42
KDM5B Q9UGL1 1/20 0.42
TSHR P16473 1/20 0.42
HDAC3 O15379 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8642939 0.84 CHRNA7 (0.47) ALDH1A1HPGDPTGS2PTGS1L3MBTL1
SCHEMBL7460234 0.83 PTGS2 (0.69) CYP2C9PTGS2PTGS1HDAC3HDAC4
SCHEMBL8642066 0.83 PTGS2 (0.47) ALDH1A1HPGDCYP1A2CYP2C9CYP2C19
SCHEMBL7466958 0.83 PTGS2 (0.55) ALDH1A1HPGDPTGS2PTGS1HDAC3
SCHEMBL8642428 0.82 CA9 (0.58) ALDH1A1MAPTMAPK1PPP1CASMN1; SMN2
SCHEMBL8642605 0.80 NPC1 (0.48) ALDH1A1HPGDCYP1A2CYP2C9CYP2C19
Dimethylamine SCHEMBL9211092 0.78 NPC1 (0.49) ALDH1A1HPGDCYP1A2CYP2C9CYP2C19
SCHEMBL15346633 0.77 ALDH1A1 (0.84) ALDH1A1HPGDCYP1A2CYP2C9CYP2C19
SCHEMBL8642612 0.77 ALDH1A1 (0.46) ALDH1A1HPGDCYP1A2CYP2C9CYP2C19
SCHEMBL8640795 0.76 KDM4C (0.50) ALDH1A1HPGDCYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0856000-A1 1,3,5-TRISUBSTITUTED PYRAZOLES FOR TREAMENT OF INFLAMMATION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-08-05 EP disclosed
WO-1997013755-A1 1,3,5-TRISUBSTITUTED PYRAZOLES FOR TREAMENT OF INFLAMMATION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-04-17 WO disclosed