SCHEMBL7469205

SCHEMBL7469205

CCOC(=O)c1ccc(N(CC(O)COc2ccc(N=Nc3ccc([N+](=O)[O-])cc3)nc2)C2CCNCC2)nc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.39
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
MAOB P27338 1/20 0.35
GAA P10253 2/20 0.35
PTPN1 P18031 1/20 0.34
PTPN6 P29350 1/20 0.34
PTPN11 Q06124 1/20 0.34
MAPT P10636 5/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KCNJ1 P48048 1/20 0.32
KCNH2 Q12809 1/20 0.32
HTT P42858 2/20 0.32
ADRB2 P07550 2/20 0.32
ADRB1 P08588 2/20 0.32
ADRB3 P13945 2/20 0.32
BCHE P06276 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7469212 0.84 MAOB (0.35) SMN1; SMN2MEN1KMT2AMAOBPTPN1
SCHEMBL7470305 0.81 MAPT (0.37) SMN1; SMN2ALDH1A1GAAMAPTNPC1
SCHEMBL7465477 0.76 MAPT (0.35) SMN1; SMN2ALDH1A1KMT2AGAAMAPT
SCHEMBL7473197 0.72 HRH3 (0.33) ALDH1A1MAPTKDM4EKCNH2ADRB2
SCHEMBL7827854 0.72 RXRA (0.36) ALDH1A1MAPTADRB2ADRB1ADRB3
SCHEMBL7468835 0.70 TLR4 (0.32) MAPT
SCHEMBL7469316 0.70 ADRB3 (0.42) MEN1KMT2AMAPTKCNH2ADRB2
SCHEMBL7460844 0.70 TLR4 (0.32) MAPT
SCHEMBL7823802 0.69 BRD4 (0.36) ALDH1A1MEN1KMT2AMAPT
SCHEMBL7822122 0.69 MAPT (0.36) SMN1; SMN2ALDH1A1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214313-A2 HETEROARYLOXY PROPANOLAMINES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI-SYNTHELABO (FR) 2002-06-19 EP disclosed
WO-2001017989-A2 HETEROARYLOXYPROPANOLAMINES AS BETA3-ADRENERGIC RECEPTOR AGONISTS SANOFI-SYNTHELABO (FR) 2001-03-15 WO disclosed