SCHEMBL7470148

SCHEMBL7470148

CCOC(=O)c1ccc(N(C2CCNCC2)C(CCO)Oc2cccc(N)c2N)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
MAOA P21397 1/20 0.34
SLC6A4 P31645 6/20 0.33
SLC6A2 P23975 5/20 0.33
SLC6A3 Q01959 4/20 0.33
CYP2D6 P10635 3/20 0.33
PTGER4 P35408 1/20 0.33
ALOX15 P16050 1/20 0.32
CHRM3 P20309 1/20 0.32
KCNH2 Q12809 1/20 0.32
RAB9A P51151 1/20 0.32
ABL1 P00519 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
RIN1 Q13671 1/20 0.32
TACR1 P25103 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7470143 0.76 MAPT (0.36) LMNACYP1A2CYP3A4MAOASLC6A4
SCHEMBL7473202 0.75 HRH3 (0.34) LMNACYP1A2CYP3A4MAOASLC6A4
SCHEMBL7473197 0.68 HRH3 (0.33) SLC6A4SLC6A2SLC6A3CYP2D6PTGER4
SCHEMBL6309219 0.64 ADRB1 (0.39) LMNACYP1A2CYP3A4MAOAALOX15
SCHEMBL4585642 0.63 LOXL2 (0.39) SLC6A4SLC6A2SLC6A3KCNH2RAB9A
SCHEMBL27574703 0.62 CA12 (0.45) LMNACYP1A2CYP3A4MAOASLC6A4
SCHEMBL15231562 0.62 ESR2 (0.51) LMNACYP1A2CYP3A4MAOARAB9A
SCHEMBL4585644 0.61 MAPT (0.40) SLC6A4SLC6A2SLC6A3KCNH2MAPT
Hydrochloric Acid SCHEMBL15231866 0.61 ESR2 (0.50) LMNACYP1A2CYP3A4MAOACYP2D6
Benzocaine SCHEMBL11645997 0.60 LMNA (0.75) LMNACYP1A2CYP3A4MAOASLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214313-A2 HETEROARYLOXY PROPANOLAMINES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI-SYNTHELABO (FR) 2002-06-19 EP disclosed
WO-2001017989-A2 HETEROARYLOXYPROPANOLAMINES AS BETA3-ADRENERGIC RECEPTOR AGONISTS SANOFI-SYNTHELABO (FR) 2001-03-15 WO disclosed