SCHEMBL7470169

SCHEMBL7470169

O=C(O)C(Cc1ccc(OCc2ccccc2)cc1)NS(=O)(=O)c1ccc(F)cc1

nearest known ligand 0.66

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPR34 Q9UPC5 2/20 0.66
MMP2 P08253 11/20 0.62
MMP9 P14780 6/20 0.62
ADAMTS4 O75173 5/20 0.62
AR P10275 1/20 0.61
MMP13 P45452 4/20 0.58
MMP14 P50281 2/20 0.58
ITGB3 P05106 1/20 0.57
ITGA2B P08514 1/20 0.57
ADAMTS5 Q9UNA0 1/20 0.57
ALDH1A1 P00352 1/20 0.57
MAPT P10636 1/20 0.57
MMP1 P03956 1/20 0.57
MMP3 P08254 1/20 0.57
MMP7 P09237 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7470160 1.00 GPR34 (0.66) GPR34MMP2MMP9ADAMTS4AR
SCHEMBL6037683 0.92 MMP2 (0.66) MMP2MMP9ADAMTS4MMP13MMP14
SCHEMBL6037682 0.92 MMP2 (0.66) MMP2MMP9ADAMTS4MMP13MMP14
SCHEMBL7468716 0.88 MMP2 (0.79) MMP2MMP9ADAMTS4MMP13ADAMTS5
SCHEMBL7460419 0.88 MMP2 (0.79) MMP2MMP9ADAMTS4MMP13ADAMTS5
SCHEMBL5189189 0.88 MMP2 (0.79) MMP2MMP9ADAMTS4MMP13ADAMTS5
SCHEMBL14602239 0.86 MMP2 (0.79) GPR34MMP2MMP9ADAMTS4AR
SCHEMBL8385428 0.86 ITGB3 (0.61) GPR34MMP2MMP9ADAMTS4MMP13
SCHEMBL8652246 0.86 ITGB3 (0.61) GPR34MMP2MMP9ADAMTS4MMP13
SCHEMBL27540161 0.84 MMP2 (0.57) MMP2MMP9ADAMTS4MMP13MMP14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0874836-B1 SULFONAMIDE INHIBITORS OF MATRIX METALLOPROTEINASES WARNER LAMBERT CO (US) 2002-10-09 EP disclosed
US-6297247-B1 Sulfonamide inhibitors of matrix metalloproteinases WARNER-LAMBERT COMPANY 2001-10-02 US disclosed
US-6153612-A Sulfonamide inhibitors of matrix metalloproteinases WARNER-LAMBERT COMPANY (US) 2000-11-28 US disclosed
US-5977141-A Sulfonamide inhibitors of matrix metalloproteinases WARNER-LAMBERT COMPANY (US) 1999-11-02 US disclosed
EP-0874836-A1 SULFONAMIDE INHIBITORS OF MATRIX METALLOPROTEINASES WARNER-LAMBERT COMPANY (US) 1998-11-04 EP disclosed
WO-1997019068-A1 SULFONAMIDE INHIBITORS OF MATRIX METALLOPROTEINASES WARNER-LAMBERT COMPANY (US) 1997-05-29 WO disclosed