SCHEMBL7470468

SCHEMBL7470468

CN(CCc1ccccc1)C1CCN(C(=O)c2ccc(-c3nc4ccccc4[nH]3)cc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 3/20 0.56
HTR2B P41595 9/20 0.54
CHEK2 O96017 2/20 0.49
MMP2 P08253 2/20 0.48
MMP13 P45452 2/20 0.48
HPGD P15428 3/20 0.47
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
KMT2A Q03164 1/20 0.47
MMP9 P14780 1/20 0.47
MMP8 P22894 1/20 0.47
HRH3 Q9Y5N1 1/20 0.46
NPC1 O15118 1/20 0.45
LMNA P02545 1/20 0.45
PKM P14618 1/20 0.45
NFKB1 P19838 1/20 0.45
RAB9A P51151 1/20 0.45
NFKB2 Q00653 1/20 0.45
RELA Q04206 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7472433 0.85 HRH4 (0.56)
Hydrochloric Acid SCHEMBL7471105 0.83 HTR2B (0.52) ATRHTR2BKDM4EALDH1A1HRH3
SCHEMBL7466231 0.80 L3MBTL3 (0.50) HTR2BHPGDALDH1A1KMT2ALMNA
Hydrochloric Acid SCHEMBL7470971 0.79 HTR2B (0.46) HTR2BCHEK2HPGDKMT2AHRH3
Hydrochloric Acid SCHEMBL7470958 0.79 HTR2B (0.46) HTR2BHPGDKMT2AHRH3NPC1
SCHEMBL9210225 0.79 CHIA (0.46) HTR2BKMT2AHRH3LMNA
SCHEMBL7465052 0.78 L3MBTL3 (0.52) KMT2ALMNA
Hydrochloric Acid SCHEMBL7476858 0.78 L3MBTL3 (0.52) KMT2ALMNA
SCHEMBL8106205 0.78 ALDH1A1 (0.56) HPGDALDH1A1KMT2ALMNA
SCHEMBL7472599 0.78 L3MBTL3 (0.52) KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0650476-B1 PERIPHERAL VASODILATING AGENT CONTAINING N-ACYLATED 4-AMINO PIPERIDINE DERIVATIVES AS ACTIVE INGREDIENTS OTSUKA PHARMA CO LTD (JP) 2002-06-26 EP disclosed
US-6136826-A AMINOPIPERIDINE COMPOUNDS SUBSTITUTED WITH ALKANOYL OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
US-5656642-A Peripheral vasodilating agent containing piperidine derivative as active ingredient OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-08-12 US disclosed
WO-1994022826-A1 PERIPHERAL VASODILATING AGENT CONTAINING N-ACYLATED 4-AMINO PIPERIDINE DERIVATIVES AS ACTIVE INGREDIENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-13 WO disclosed