SCHEMBL7470579

SCHEMBL7470579

COc1nc2cc(Cl)c(Cl)c(CSCc3ccccc3)c2nc1OC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 2/20 0.34
SMN1; SMN2 Q16637 4/20 0.34
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
KMT2A Q03164 2/20 0.34
MAPT P10636 2/20 0.34
ALDH1A1 P00352 2/20 0.34
HPGD P15428 2/20 0.34
KDM4E B2RXH2 1/20 0.34
TP53 P04637 1/20 0.34
GAA P10253 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CYP2E1 P05181 1/20 0.34
CYP2C8 P10632 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7468650 0.80 HRH4 (0.34) PTGESNQO2
SCHEMBL7468298 0.79 KMT2A (0.37) PTGESNPC1RAB9AKMT2AALDH1A1
SCHEMBL7466499 0.74 HRH4 (0.35) PTGESNQO2
SCHEMBL8784394 0.74 HRH4 (0.35) PTGESNQO2
SCHEMBL8784365 0.72 HRH4 (0.34) PTGESALDH1A1KDM4ENQO2
SCHEMBL8784616 0.70 TLR8 (0.35) PTGESALDH1A1TDP1NQO2
SCHEMBL7467268 0.70 GLP1R (0.34) PTGESSMN1; SMN2NQO2
SCHEMBL7470559 0.69 HRH4 (0.32) PTGES
SCHEMBL7473964 0.68 HRH4 (0.39) PTGESKMT2ANR1I3MEN1NQO2
SCHEMBL8647402 0.68 PTGES (0.30) PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0783495-B1 QUINOXALINE DERIVATIVES USEFUL IN THERAPY PFIZER LTD (GB) 2002-02-27 EP disclosed
US-5852016-A Quinoxaline derivatives useful in therapy PFIZER INC. (US) 1998-12-22 US disclosed
EP-0783495-A1 QUINOXALINE DERIVATIVES USEFUL IN THERAPY Pfizer Limited (GB) 1997-07-16 EP disclosed
WO-1996009295-A1 QUINOXALINE DERIVATIVES USEFUL IN THERAPY PFIZER LIMITED (GB) 1996-03-28 WO disclosed